SCHEMBL6987858

SCHEMBL6987858

CN(Cc1ccc(Cl)cc1)C(=O)c1c[nH]c2c(I)cc(CC3CCOCC3)cc2c1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
HPGD P15428 2/20 0.42
GAA P10253 2/20 0.42
KDM4E B2RXH2 1/20 0.42
GLA P06280 1/20 0.42
MAPK14 Q16539 1/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TP53 P04637 2/20 0.34
MAPT P10636 1/20 0.34
POLB P06746 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
PDE4B Q07343 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
THRB P10828 2/20 0.33
NPC1 O15118 1/20 0.33
HSP90AA1 P07900 2/20 0.33
P2RX7 Q99572 2/20 0.33
USP2 O75604 1/20 0.33
GABRA1 P14867 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6668158 0.86 ALDH1A1 (0.54) ALDH1A1HPGDGAAKDM4EGLA
SCHEMBL6984758 0.85 ALDH1A1 (0.47) ALDH1A1HPGDGAAKDM4EGLA
SCHEMBL6989961 0.84 ALDH1A1 (0.38) ALDH1A1HPGDGAAKDM4EGLA
SCHEMBL6988955 0.84 ALDH1A1 (0.38) ALDH1A1HPGDGAAKDM4EGLA
SCHEMBL6987501 0.84 ALDH1A1 (0.41) ALDH1A1HPGDGAAKDM4EGLA
SCHEMBL7844071 0.78 NPC1 (0.43) ALDH1A1HPGDGAAKDM4EGLA
SCHEMBL7846837 0.74 GAA (0.43) ALDH1A1HPGDGAAKDM4EGLA
SCHEMBL6673044 0.74 ALDH1A1 (0.61) ALDH1A1HPGDGAAKDM4EGLA
SCHEMBL6672672 0.73 NR1H4 (0.34) MAPK14SMN1; SMN2NPC1HSP90AA1P2RX7
SCHEMBL6667531 0.73 NR1H4 (0.34) MAPK14SMN1; SMN2NPC1HSP90AA1P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1363887-A1 SUBSTITUTED QUINOLINECARBOXAMIDES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 2003-11-26 EP disclosed
WO-2002070487-A1 SUBSTITUTED QUINOLINECARBOXAMIDES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 2002-09-12 WO disclosed