SCHEMBL6988596

SCHEMBL6988596

Cc1ccc2c(c1)Nc1sc3cc(F)ccc3c1C(=O)N2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK1G1 Q9HCP0 1/20 0.41
G6PD P11413 2/20 0.38
PMM2 O15305 2/20 0.38
MPI P34949 2/20 0.38
PHOSPHO1 Q8TCT1 2/20 0.38
KAT2B Q92831 1/20 0.38
ALDH1A1 P00352 2/20 0.37
MAPT P10636 2/20 0.37
NPC1 O15118 1/20 0.37
CYP1A2 P05177 1/20 0.37
GAA P10253 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
RAB9A P51151 1/20 0.37
MCL1 Q07820 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ROS1 P08922 1/20 0.37
CDK5 Q00535 1/20 0.37
ACVR1 Q04771 1/20 0.37
LRRK2 Q5S007 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6998266 0.95 CSNK1G1 (0.38) CSNK1G1G6PDPMM2MPIPHOSPHO1
SCHEMBL6998917 0.91 CSNK1G1 (0.46) CSNK1G1ALDH1A1MAPTNPC1CYP1A2
SCHEMBL6990964 0.91 MAPT (0.40) MPIALDH1A1MAPTCYP1A2CYP2C19
SCHEMBL6993139 0.88 CSNK1G1 (0.38) CSNK1G1G6PDPMM2MPIPHOSPHO1
SCHEMBL6997151 0.85 CCNE2 (0.40) G6PDMPIPHOSPHO1ALDH1A1MAPT
SCHEMBL6992702 0.84 TGM2 (0.37) ALDH1A1MAPTCDK5LRRK2ESR1
SCHEMBL6998420 0.83 CSNK1G1 (0.50) CSNK1G1PMM2MPIPHOSPHO1ALDH1A1
SCHEMBL6994996 0.83 CSNK1G1 (0.50) CSNK1G1PMM2MPIPHOSPHO1ALDH1A1
SCHEMBL6992029 0.83 ACVR1 (0.48) CSNK1G1ALDH1A1MAPTNPC1CYP1A2
SCHEMBL6994334 0.82 MDM2 (0.42) PMM2MPIPHOSPHO1ALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1016664-B1 FUSED THIOPHENE COMPOUNDS AND MEDICINAL USE THEREOF MITSUBISHI PHARMA CORP (JP) 2003-07-02 EP claimed
US-20020042411-A1 Condensed thiophene compounds and pharmaceutical use thereof MITSUBISHI PHARMA CORPORATION (JP) 2002-04-11 US claimed
US-6271225-B1 PSYCHOLOGICAL DISORDERS WELFIDE CORPORATION (JP) 2001-08-07 US claimed
EP-1016664-A1 FUSED THIOPHENE COMPOUNDS AND MEDICINAL USE THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 2000-07-05 EP claimed
EP-1016664-B1 FUSED THIOPHENE COMPOUNDS AND MEDICINAL USE THEREOF MITSUBISHI PHARMA CORP (JP) 2003-07-02 EP disclosed
US-6455521-B1 PSYCHOLOGICAL DISORDERS; SIDE EFFECT REDUCTION MITSUBISHI PHARMA CORPORATION (JP) 2002-09-24 US disclosed
US-20020042411-A1 Condensed thiophene compounds and pharmaceutical use thereof MITSUBISHI PHARMA CORPORATION (JP) 2002-04-11 US disclosed
US-6271225-B1 PSYCHOLOGICAL DISORDERS WELFIDE CORPORATION (JP) 2001-08-07 US disclosed
EP-1016664-A1 FUSED THIOPHENE COMPOUNDS AND MEDICINAL USE THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 2000-07-05 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020042411-A1 Condensed thiophene compounds and pharmaceutical use thereof ACIN1, ACHE, TPMT CSNK1G1 1141/4885G6PD 169/4885PMM2 315/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.