SCHEMBL6989802

SCHEMBL6989802

COc1ccc(C(C=O)c2ccc(Cl)c(Cl)c2)cc1OC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.44
AKR1C2 P52895 1/20 0.44
ALDH1A1 P00352 1/20 0.42
TSHR P16473 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
GAA P10253 1/20 0.42
TNF P01375 2/20 0.41
MAPT P10636 2/20 0.41
TP53 P04637 1/20 0.41
ACHE P22303 2/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
LMNA P02545 1/20 0.40
PPARG P37231 1/20 0.40
PPARD Q03181 1/20 0.40
PPARA Q07869 1/20 0.40
RAD51 Q06609 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6994425 0.81 NPC1 (0.38) AKR1C3AKR1C2ALDH1A1SMN1; SMN2GAA
SCHEMBL1515750 0.81 L3MBTL1 (0.53) ALDH1A1TSHRGAATNFMAPT
SCHEMBL5877045 0.81 L3MBTL1 (0.53) ALDH1A1TSHRGAATNFMAPT
SCHEMBL3944811 0.79 NQO2 (0.46) ALDH1A1TSHRGAAACHECA1
SCHEMBL6508159 0.78 ALDH1A1 (0.47) ALDH1A1TSHRSMN1; SMN2GAAMAPT
SCHEMBL1010039 0.77 HSP90AA1 (0.41) ALDH1A1TSHRSMN1; SMN2GAATNF
SCHEMBL6988715 0.77 ALDH1A1 (0.45) ALDH1A1GAAMAPTLMNAKMT2A
SCHEMBL8800434 0.77 CYP1A1 (0.38) ALDH1A1TSHRSMN1; SMN2GAATP53
SCHEMBL1515724 0.75 IDO1 (0.49) ALDH1A1CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL17802349 0.75 IDO1 (0.49) ALDH1A1CYP3A4CYP2D6SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347967-A1 NOVEL BENZAZEPINES AND RELATED HETEROCYCLIC DERIVATIVES WHICH ARE USEFUL AS OREXIN RECEPTOR ANTAGONISTS Actelion Pharmaceuticals Ltd. (CH) 2003-10-01 EP disclosed
WO-2002051838-A1 NOVEL BENZAZEPINES AND RELATED HETEROCYCLIC DERIVATIVES WHICH ARE USEFUL AS OREXIN RECEPTOR ANTAGONISTS ACTELION PHARMACEUTICALS LTD. (CH) 2002-07-04 WO disclosed