SCHEMBL6991287

SCHEMBL6991287

CC1=C(N)Nc2cc(CNCc3cccc([N+](=O)[O-])c3)ccc2O1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.44
MEN1 O00255 3/20 0.44
MAPT P10636 3/20 0.44
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C19 P33261 1/20 0.42
PARP1 P09874 2/20 0.41
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
ALDH1A1 P00352 2/20 0.40
TDP1 Q9NUW8 1/20 0.39
POLB P06746 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRK1 P41145 1/20 0.39
EGFR P00533 1/20 0.39
PTPN1 P18031 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6997432 0.99 KMT2A (0.44) KMT2AMEN1MAPTCYP1A2CYP3A4
SCHEMBL6995764 0.90 CHRM2 (0.41) KMT2AMEN1MAPTPARP1ALDH1A1
Hydrochloric Acid SCHEMBL6992777 0.89 CHRM2 (0.40) KMT2AMEN1MAPTPARP1ALDH1A1
Hydrochloric Acid SCHEMBL7713373 0.82 PARP1 (0.53) KMT2AMEN1PARP1ALDH1A1TDP1
SCHEMBL6998348 0.81 KDM4E (0.45) KMT2AMEN1CYP1A2CYP2C19PARP1
SCHEMBL7002250 0.81 PARP1 (0.42) PARP1OPRM1OPRK1
SCHEMBL7002470 0.81 PARP1 (0.42) CYP1A2CYP3A4CYP2C19PARP1
Hydrochloric Acid SCHEMBL6994806 0.81 KDM4E (0.44) KMT2AMEN1CYP1A2CYP2C19PARP1
Hydrochloric Acid SCHEMBL7001196 0.80 PARP1 (0.41) PARP1
Hydrochloric Acid SCHEMBL6996848 0.80 PARP1 (0.41) CYP1A2CYP3A4CYP2C19PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015437-B1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN PHARMACEUTICALS SCHERING AG (DE) 2003-12-03 EP claimed