SCHEMBL7002250

SCHEMBL7002250

CC1=C(N)Nc2cc(CNCc3cccc(F)c3)ccc2O1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.42
SCN8A Q9UQD0 1/20 0.39
NOS1 P29475 3/20 0.39
PDGFRB P09619 1/20 0.37
KDR P35968 1/20 0.37
ATM Q13315 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MPO P05164 2/20 0.36
NOS3 P29474 1/20 0.35
NOS2 P35228 1/20 0.35
MAPK1 P28482 1/20 0.35
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7001196 0.99 PARP1 (0.41) PARP1SCN8ANOS1PDGFRBKDR
SCHEMBL6994032 0.89 LMNA (0.42) PARP1PDGFRBKDRL3MBTL1MAPK1
Hydrochloric Acid SCHEMBL6996205 0.88 PARP1 (0.41) PARP1PDGFRBKDRMAPK1
Hydrochloric Acid SCHEMBL7713373 0.86 PARP1 (0.53) PARP1PDGFRBKDRATM
SCHEMBL7002470 0.86 PARP1 (0.42) PARP1NOS1PDGFRBKDRNOS3
Hydrochloric Acid SCHEMBL6996848 0.85 PARP1 (0.41) PARP1NOS1PDGFRBKDRNOS3
Hydrochloric Acid SCHEMBL6999647 0.84 SCN8A (0.42) PARP1SCN8ANOS1NOS2
Hydrochloric Acid SCHEMBL6310054 0.84 PARP1 (0.42) PARP1
SCHEMBL7002617 0.84 PARP1 (0.41) PARP1SCN8APDGFRBKDRMAPK1
SCHEMBL6998348 0.84 KDM4E (0.45) PARP1SCN8APDGFRBKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015437-B1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN PHARMACEUTICALS SCHERING AG (DE) 2003-12-03 EP claimed