SCHEMBL7002470

SCHEMBL7002470

CC1=C(N)Nc2cc(CNCc3cccc(Cl)c3)ccc2O1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.42
CHRM2 P08172 1/20 0.42
HDAC1 Q13547 1/20 0.41
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
NOS3 P29474 2/20 0.39
NOS1 P29475 2/20 0.39
NOS2 P35228 2/20 0.39
PDGFRB P09619 1/20 0.38
KDR P35968 1/20 0.38
LMNA P02545 1/20 0.36
CXCR4 P61073 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6996848 0.99 PARP1 (0.41) PARP1CHRM2HDAC1CYP1A2CYP3A4
SCHEMBL6993345 0.89 PARP1 (0.42) PARP1CHRM2LMNA
Hydrochloric Acid SCHEMBL6996685 0.88 PARP1 (0.41) PARP1CHRM2LMNA
Hydrochloric Acid SCHEMBL7713373 0.86 PARP1 (0.53) PARP1PDGFRBKDR
SCHEMBL7002250 0.86 PARP1 (0.42) PARP1NOS3NOS1NOS2PDGFRB
SCHEMBL6993016 0.85 L3MBTL1 (0.45) PARP1CYP1A2CYP2D6CYP2C19
SCHEMBL6996665 0.85 HTT (0.39) PARP1CYP1A2CYP3A4CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL7001196 0.85 PARP1 (0.41) PARP1NOS3NOS1NOS2PDGFRB
Hydrochloric Acid SCHEMBL6990749 0.84 L3MBTL1 (0.44) PARP1CYP1A2CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL6998295 0.84 HTT (0.41) PARP1CYP1A2CYP3A4CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015437-B1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN PHARMACEUTICALS SCHERING AG (DE) 2003-12-03 EP claimed