SCHEMBL6991868

SCHEMBL6991868

O=C(NC(Cc1ccc(Cl)c(Cl)c1)C(=O)NC12CCCC1OCC2=O)c1ccc(OC(F)F)cc1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSL P07711 11/20 0.39
KLKB1 P03952 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
IDO1 P14902 1/20 0.37
KMT2A Q03164 1/20 0.37
SSTR3 P32745 2/20 0.35
CTSB P07858 1/20 0.35
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
SRC P12931 1/20 0.35
ZAP70 P43403 1/20 0.35
PRSS1 P07477 1/20 0.35
PRSS2 P07478 1/20 0.35
PRSS3 P35030 1/20 0.35
TPSAB1 Q15661 1/20 0.35
UTS2R Q9UKP6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6300424 0.92 IDO1 (0.44) CTSLIDO1KMT2ACTSBCTSS
SCHEMBL6701575 0.90 TRPV1 (0.44) CTSLKLKB1CYP2D6CYP2C9
SCHEMBL6300527 0.90 CTSL (0.38) CTSLIDO1KMT2ACTSBCTSS
SCHEMBL6300604 0.89 CTSL (0.38) CTSLIDO1KMT2ACTSBCTSS
SCHEMBL6294295 0.88 CTSL (0.40) CTSLCYP2D6CYP2C9SSTR3
SCHEMBL6295728 0.88 CTSL (0.36) CTSLKLKB1IDO1KMT2ASSTR3
SCHEMBL6702836 0.88 CTSL (0.41) CTSLKLKB1CYP2D6CYP2C9CTSB
SCHEMBL6699255 0.87 CTSL (0.40) CTSLKLKB1CYP2D6CYP2C9SSTR3
SCHEMBL6695685 0.86 CTSB (0.45) CTSLKLKB1CYP2D6CYP2C9KMT2A
SCHEMBL6699096 0.83 CTSL (0.45) CTSLIDO1KMT2ACTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1358176-A2 INHIBITORS OF CRUZIPAIN AND OTHER CYSTEINE PROTEASES Amura Therapeutics Limited (GB) 2003-11-05 EP disclosed
WO-2002057246-A2 INHIBITORS OF CRUZIPAIN AND OTHER CYSTEINE PROTEASES AMURA THERAPEUTICS LIMITED (GB) 2002-07-25 WO disclosed