SCHEMBL6992026

SCHEMBL6992026

Cc1ccc(NC(=O)c2c(Br)sc3c2CCCC3)c(O)c1

nearest known ligand 0.67

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.67
THRB P10828 1/20 0.67
SMN1; SMN2 Q16637 4/20 0.46
GAA P10253 2/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
TP53 P04637 5/20 0.46
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
FLT3 P36888 2/20 0.46
ANO1 Q5XXA6 4/20 0.45
ANO2 Q9NQ90 2/20 0.45
LMNA P02545 1/20 0.45
POLB P06746 1/20 0.44
BLM P54132 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7000741 0.88 MAPT (0.67) MAPTTHRBSMN1; SMN2TP53KMT2A
SCHEMBL6995066 0.86 MAPT (0.55) MAPTTHRBNPC1RAB9ATP53
SCHEMBL6993062 0.83 MAPT (0.59) MAPTTHRBSMN1; SMN2NPC1RAB9A
SCHEMBL6998812 0.77 MAPT (0.55) MAPTTHRBGAANPC1RAB9A
SCHEMBL6991198 0.76 MAPT (0.59) MAPTTHRBSMN1; SMN2NPC1RAB9A
SCHEMBL6995125 0.71 RAB9A (0.53) MAPTSMN1; SMN2GAANPC1RAB9A
SCHEMBL17224032 0.71 RAB9A (0.53) MAPTSMN1; SMN2GAANPC1RAB9A
SCHEMBL12172944 0.71 GAA (0.56) MAPTSMN1; SMN2GAANPC1RAB9A
SCHEMBL7217418 0.69 CYP1A2 (0.68) MAPTTHRBSMN1; SMN2GAATP53
SCHEMBL12443269 0.69 ANO1 (0.75) MAPTSMN1; SMN2TP53ANO1ANO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1016664-B1 FUSED THIOPHENE COMPOUNDS AND MEDICINAL USE THEREOF MITSUBISHI PHARMA CORP (JP) 2003-07-02 EP disclosed
US-6455521-B1 PSYCHOLOGICAL DISORDERS; SIDE EFFECT REDUCTION MITSUBISHI PHARMA CORPORATION (JP) 2002-09-24 US disclosed
US-20020042411-A1 Condensed thiophene compounds and pharmaceutical use thereof MITSUBISHI PHARMA CORPORATION (JP) 2002-04-11 US disclosed
US-6271225-B1 PSYCHOLOGICAL DISORDERS WELFIDE CORPORATION (JP) 2001-08-07 US disclosed
EP-1016664-A1 FUSED THIOPHENE COMPOUNDS AND MEDICINAL USE THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 2000-07-05 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020042411-A1 Condensed thiophene compounds and pharmaceutical use thereof ACIN1, ACHE, TPMT MAPT 15/4885THRB 1692/4885SMN1; SMN2 1349/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.