SCHEMBL6992860

SCHEMBL6992860

COC(=O)C(Cc1ccc(I)cc1)N(C)C(=O)OC(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 1/20 0.41
REN P00797 1/20 0.39
AAK1 Q2M2I8 2/20 0.38
MMP13 P45452 1/20 0.38
ITGA4 P13612 1/20 0.37
ITGB7 P26010 1/20 0.37
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
KLK5 Q9Y337 2/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
PTPRB P23467 1/20 0.33
APEX1 P27695 1/20 0.33
PMP22 Q01453 1/20 0.33
P2RX7 Q99572 1/20 0.33
ABCB1 P08183 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20422635 0.88 ESR1 (0.49) ADORA1RENAAK1MMP13ITGA4
SCHEMBL20422634 0.88 ESR1 (0.49) ADORA1RENAAK1MMP13ITGA4
SCHEMBL15702033 0.88 ITGA4 (0.38) ADORA1ITGA4ITGB7ESR1ESR2
SCHEMBL3638571 0.87 LDHA (0.46) ADORA1RENMMP13ITGA4ITGB7
SCHEMBL8362444 0.87 ADORA1 (0.51) ADORA1RENAAK1MMP13ITGA4
SCHEMBL23279486 0.87 MEN1 (0.41) ADORA1RENAAK1MMP13ITGA4
SCHEMBL18256513 0.87 MEN1 (0.41) ADORA1RENAAK1MMP13ITGA4
SCHEMBL7906205 0.87 ADORA1 (0.44) ADORA1RENAAK1MMP13ITGA4
SCHEMBL8362441 0.87 ADORA1 (0.51) ADORA1RENAAK1MMP13ITGA4
SCHEMBL1325201 0.87 MMP13 (0.39) ADORA1RENAAK1MMP13ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8492345-B2 Cyclic peptide antitumor agents NORTHWESTERN UNIVERSITY (US) 2013-07-23 US disclosed
US-20120122799-A1 CYCLIC PEPTIDE ANTITUMOR AGENTS NORTHWESTERN UNIVERSITY (US) 2012-05-17 US disclosed
US-8058244-B2 Cyclic peptide antitumor agents NORTHWESTERN UNIVERSITY (US) 2011-11-15 US disclosed
US-8058244-B2 Cyclic peptide antitumor agents NORTHWESTERN UNIVERSITY (US) 2011-11-15 US disclosed
US-20100204088-A1 Cyclic Peptide Antitumor Agents SILVERMAN RICHARD B 2010-08-12 US disclosed
US-20100204088-A1 Cyclic Peptide Antitumor Agents SILVERMAN RICHARD B 2010-08-12 US disclosed
US-7709443-B2 For treatment of human melanoma, pancreatic, breast, prostate cancer cells NORTHWESTERN UNIVERSITY (US) 2010-05-04 US disclosed
US-7709443-B2 For treatment of human melanoma, pancreatic, breast, prostate cancer cells NORTHWESTERN UNIVERSITY (US) 2010-05-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100204088-A1 Cyclic Peptide Antitumor Agents VIP, IAPP, NGLY1 ADORA1 4669/4885REN 4100/4885AAK1 3219/4885
US-20120122799-A1 CYCLIC PEPTIDE ANTITUMOR AGENTS VIP, IAPP, NGLY1 ADORA1 4669/4885REN 4100/4885AAK1 3219/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.