SCHEMBL6993246

SCHEMBL6993246

CCn1ccc2c1C(=O)N(CCCN1CCN(c3ccc(F)cc3)CC1)CC/C2=N/O

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.45
LMNA P02545 1/20 0.45
MAPK1 P28482 1/20 0.45
DRD3 P35462 5/20 0.42
DRD2 P14416 2/20 0.41
DRD4 P21917 1/20 0.39
DRD1 P21728 1/20 0.39
SIGMAR1 Q99720 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6993251 1.00 KDM4E (0.45) KDM4ELMNAMAPK1DRD3DRD2
SCHEMBL6993431 0.91 HTR1A (0.46) DRD3DRD2DRD4DRD1
SCHEMBL6993434 0.91 HTR1A (0.46) DRD3DRD2DRD4DRD1
SCHEMBL6989852 0.90 KDM4E (0.47) KDM4ELMNAMAPK1DRD3DRD2
SCHEMBL6989849 0.90 KDM4E (0.47) KDM4ELMNAMAPK1DRD3DRD2
SCHEMBL6993564 0.88 KDM4E (0.46) KDM4ELMNAMAPK1DRD3DRD2
SCHEMBL6987644 0.84 DRD2 (0.48) KDM4ELMNAMAPK1DRD3DRD2
SCHEMBL6768552 0.84 KDM4E (0.47) KDM4ELMNAMAPK1DRD3DRD2
SCHEMBL6768554 0.84 KDM4E (0.47) KDM4ELMNAMAPK1DRD3DRD2
SCHEMBL6987645 0.84 DRD2 (0.48) KDM4ELMNAMAPK1DRD3DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0557526-B1 PYRROLOAZEPINE COMPOUND SUNTORY LTD (JP) 2003-04-02 EP disclosed
US-5399557-A Cardiovascular disorders SUNTORY LIMITED (JP) 1995-03-21 US disclosed
EP-0557526-A1 PYRROLOAZEPINE COMPOUND SUNTORY LIMITED (JP) 1993-09-01 EP disclosed