SCHEMBL6993286

SCHEMBL6993286

NC(=O)c1nc2cc(CO)ccc2s1.NCc1cccc(N(CC(=O)O)C(=O)c2ccccc2)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.37
RAB9A P51151 5/20 0.37
HPGD P15428 3/20 0.37
NFKB1 P19838 2/20 0.37
NFKB2 Q00653 2/20 0.37
RELA Q04206 2/20 0.37
STAT1 P42224 1/20 0.37
F2 P00734 3/20 0.37
KDM4E B2RXH2 1/20 0.36
HSD17B10 Q99714 1/20 0.35
ADRA2C P18825 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
CYP3A4 P08684 1/20 0.33
LTB4R2 Q9NPC1 1/20 0.32
KMT2A Q03164 1/20 0.32
GFER P55789 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
MCL1 Q07820 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5208572 0.95 F2 (0.40) NPC1RAB9AHPGDNFKB1NFKB2
SCHEMBL6996710 0.90 NPC1 (0.43) NPC1RAB9AHPGDNFKB1NFKB2
SCHEMBL5208349 0.88 F2 (0.40) NPC1F2ADRA2CCYP3A4MAPT
SCHEMBL5207728 0.84 NPC1 (0.43) NPC1RAB9AHPGDNFKB1NFKB2
Trifluoroacetic Acid SCHEMBL5211180 0.80 NPC1 (0.39) NPC1RAB9AHPGDF2ADRA2C
SCHEMBL6991435 0.80 F2 (0.35) NPC1RAB9AF2KDM4EADRA2C
SCHEMBL7432548 0.79 TP53 (0.41) NPC1RAB9AHPGDF2KDM4E
SCHEMBL6988918 0.78 ADRA2C (0.52) NPC1RAB9AADRA2CKMT2AGAA
Trifluoroacetic Acid SCHEMBL5210737 0.77 F2 (0.38) F2ADRA2CKMT2AMAPTPKM
Trifluoroacetic Acid SCHEMBL7432339 0.77 LMNA (0.37) NPC1RAB9AHPGDF2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1343561-A1 SERINE PROTEASE INHIBITORS Tularik Limited (GB) 2003-09-17 EP disclosed
WO-2002047762-A1 SERINE PROTEASE INHIBITORS TULARIK LIMITED (GB) 2002-06-20 WO disclosed