SCHEMBL6991435

SCHEMBL6991435

NC(=O)c1nc2c(s1)CCCC2.NCc1cccc(N(CC(=O)O)C(=O)c2ccccc2)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2 P00734 1/20 0.35
RAB9A P51151 5/20 0.35
MAPT P10636 5/20 0.35
SMN1; SMN2 Q16637 4/20 0.35
NPC1 O15118 4/20 0.35
PKM P14618 2/20 0.35
ALDH1A1 P00352 8/20 0.35
POLB P06746 3/20 0.35
ADRA2C P18825 1/20 0.35
KMT2A Q03164 3/20 0.35
TP53 P04637 2/20 0.35
MEN1 O00255 2/20 0.35
LMNA P02545 4/20 0.34
SLC12A2 P55011 1/20 0.34
SLC12A5 Q9H2X9 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
MITF O75030 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5210132 0.95 F2 (0.39) F2RAB9AMAPTSMN1; SMN2NPC1
Hydrochloric Acid SCHEMBL5208877 0.85 PIK3CA (0.35) RAB9AMAPTSMN1; SMN2NPC1PKM
Trifluoroacetic Acid SCHEMBL6999298 0.83 HRH2 (0.37) RAB9AMAPTSMN1; SMN2NPC1ALDH1A1
Trifluoroacetic Acid SCHEMBL6993355 0.83 OPRM1 (0.33) F2PKMKMT2AMEN1LMNA
Trifluoroacetic Acid SCHEMBL5203620 0.82 PIK3CA (0.33) RAB9AMAPTSMN1; SMN2NPC1PKM
SCHEMBL6996710 0.81 NPC1 (0.43) F2RAB9AMAPTSMN1; SMN2NPC1
Trifluoroacetic Acid SCHEMBL6996192 0.81 HRH2 (0.34) RAB9AMAPTPKMALDH1A1KMT2A
Trifluoroacetic Acid SCHEMBL5208291 0.80 MAPT (0.33) F2RAB9AMAPTSMN1; SMN2NPC1
Trifluoroacetic Acid SCHEMBL6994655 0.80 OPRD1 (0.34) PKMKMT2AMEN1OPRM1OPRD1
SCHEMBL6993286 0.80 NPC1 (0.37) F2RAB9AMAPTSMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1343561-A1 SERINE PROTEASE INHIBITORS Tularik Limited (GB) 2003-09-17 EP disclosed
WO-2002047762-A1 SERINE PROTEASE INHIBITORS TULARIK LIMITED (GB) 2002-06-20 WO disclosed