SCHEMBL6993377

SCHEMBL6993377

O=C(COc1ncccn1)OC(=O)C(F)(F)F

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.31
NPC1 O15118 1/20 0.31
TSHR P16473 1/20 0.31
RXRA P19793 1/20 0.30
GRIN1 Q05586 1/20 0.30
GRIN2B Q13224 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11354741 0.76 ALOX15 (0.53) NPC1
SCHEMBL2413467 0.75 MAPT (0.45)
Trifluoroacetic Acid SCHEMBL6993373 0.75 ALOX15 (0.42) TSHR
SCHEMBL6990825 0.74 KMT2A (0.34) TDP1NPC1TSHRRXRAGRIN1
SCHEMBL6496575 0.71 ALDH1A1 (0.41) NPC1TSHR
SCHEMBL16756469 0.71 SMARCA2 (0.37)
SCHEMBL315714 0.69 KDM4E (0.50) TSHR
SCHEMBL1280673 0.69 ALOX15 (0.52) TDP1
SCHEMBL5859013 0.67 MAPT (0.49) TDP1
SCHEMBL4658964 0.67 CES1 (0.47) TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1476436-A Novel compounds for use as HIV protease inhibitors - 2004-02-18 CN disclosed
EP-1339692-A1 NOVEL COMPOUNDS FOR USE AS HIV PROTEASE INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2003-09-03 EP disclosed
US-6472404-B1 HIV protease inhibitors HOFFMANN-LA ROCHE INC. 2002-10-29 US disclosed
WO-2002042277-A1 NOVEL COMPOUNDS FOR USE AS HIV PROTEASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2002-05-30 WO disclosed