SCHEMBL6993447

SCHEMBL6993447

CCn1ccc2c1C(=O)N(CCCCl)CC/C2=N/O

nearest known ligand 0.32

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.32
HPGD P15428 4/20 0.32
MEN1 O00255 2/20 0.32
POLB P06746 2/20 0.32
MAPT P10636 2/20 0.32
BLM P54132 2/20 0.32
KMT2A Q03164 2/20 0.32
MCL1 Q07820 2/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
KDM4E B2RXH2 2/20 0.32
LMNA P02545 1/20 0.31
ALOX12 P18054 1/20 0.31
NPC1 O15118 2/20 0.30
RAB9A P51151 2/20 0.30
SMN1; SMN2 Q16637 2/20 0.30
HSD17B10 Q99714 2/20 0.30
GRM5 P41594 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6993449 1.00 ALDH1A1 (0.32) ALDH1A1HPGDMEN1POLBMAPT
SCHEMBL9037511 0.88 NPC1 (0.35) ALDH1A1HPGDKDM4ELMNANPC1
SCHEMBL9039600 0.88 HTT (0.31)
SCHEMBL6997468 0.87 KDM4E (0.31) ALDH1A1HPGDMEN1POLBMAPT
SCHEMBL6997471 0.87 KDM4E (0.31) ALDH1A1HPGDMEN1POLBMAPT
SCHEMBL9040156 0.87 GRM5 (0.32) GRM5
SCHEMBL6994951 0.84 PTPN1 (0.36) ALDH1A1HPGDMEN1POLBMAPT
SCHEMBL9039276 0.82
SCHEMBL6993434 0.81 HTR1A (0.46)
SCHEMBL6993431 0.81 HTR1A (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0557526-B1 PYRROLOAZEPINE COMPOUND SUNTORY LTD (JP) 2003-04-02 EP disclosed
US-5399557-A Cardiovascular disorders SUNTORY LIMITED (JP) 1995-03-21 US disclosed
EP-0557526-A1 PYRROLOAZEPINE COMPOUND SUNTORY LIMITED (JP) 1993-09-01 EP disclosed