SCHEMBL6993752

SCHEMBL6993752

c1ccc2[nH]c(CC3=NCCCN3)nc2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.53
BCHE P06276 1/20 0.48
DDAH1 O94760 1/20 0.47
POLB P06746 1/20 0.47
LMNA P02545 3/20 0.47
HTT P42858 2/20 0.47
TSHR P16473 2/20 0.47
PKM P14618 2/20 0.47
KRAS P01116 1/20 0.45
GRIN1 Q05586 1/20 0.45
GRIN2B Q13224 1/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
EGFR P00533 1/20 0.44
ERBB2 P04626 1/20 0.44
MAPT P10636 1/20 0.44
HKDC1 Q2TB90 1/20 0.44
CYP1A2 P05177 1/20 0.43
ADRA2A P08913 1/20 0.43
CYP2D6 P10635 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7000055 0.96 GAA (0.51) GAABCHEDDAH1POLBLMNA
SCHEMBL6992236 0.91 GAA (0.55) GAABCHEDDAH1POLBLMNA
SCHEMBL230024 0.76 GAA (0.78) GAABCHEDDAH1POLBLMNA
SCHEMBL6998141 0.74 GAA (0.49) GAABCHEDDAH1POLBLMNA
SCHEMBL6994270 0.72 DDAH1 (0.49) GAABCHEDDAH1POLBLMNA
SCHEMBL11597510 0.72 TAAR1 (0.79) GAALMNATSHRCYP1A2ADRA2A
Hydrochloric Acid SCHEMBL7230476 0.71 DDAH1 (0.48) GAABCHEDDAH1POLBLMNA
Iodomethane SCHEMBL27491515 0.71 GAA (0.70) GAABCHEDDAH1POLBLMNA
SCHEMBL6993819 0.70 DDAH1 (0.54) GAABCHEDDAH1POLBLMNA
SCHEMBL6994631 0.70 GAA (0.51) GAADDAH1POLBLMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1189889-B1 COMPOSITIONS AND METHODS FOR INHIBITING CELL DEATH ELAN PHARMA INT LTD (IE) 2003-12-17 EP claimed
EP-1189889-B1 COMPOSITIONS AND METHODS FOR INHIBITING CELL DEATH ELAN PHARMA INT LTD (IE) 2003-12-17 EP disclosed
US-6541486-B1 Used for treating ischemia, such as results from stroke or myocardial infarction, trauma, neurodegeneration, and inflammation. ELAN PHARMA INTERNATIONAL LTD. (IE) 2003-04-01 US disclosed