SCHEMBL6995017

SCHEMBL6995017

O=C1OC2(CCC2)C(OS(=O)(=O)C(F)(F)F)=C1c1ccccc1

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.32
SIGMAR1 Q99720 1/20 0.32
PTGS1 P23219 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.31
PDE4B Q07343 1/20 0.31
KMT2A Q03164 1/20 0.30
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30
BACE1 P56817 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8003087 0.74 CYSLTR1 (0.35)
SCHEMBL1420100 0.74 CYSLTR1 (0.46)
SCHEMBL6997284 0.69 SIGMAR1 (0.38) PTGS2SIGMAR1PTGS1SMN1; SMN2KMT2A
SCHEMBL17314725 0.67 PTGS2 (0.38) PTGS2PTGS1PDE4BKMT2AADORA2A
SCHEMBL13880121 0.67 HRH3 (0.39) SIGMAR1
SCHEMBL6993378 0.66 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL6989032 0.66 PTGS2 (0.54) PTGS2PTGS1
Biphenyl SCHEMBL28551760 0.64 CA1 (0.53) KMT2AADORA2AADORA1
SCHEMBL6991312 0.63 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL6986739 0.63 PTGS2 (0.54) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0799218-B1 DIARYL-2-(5H)-FURANONES AS COX-2 INHIBITORS MERCK FROSST CANADA INC (CA) 2003-02-19 EP disclosed
US-6222048-B1 AS ANTIINFLAMMATORY, ANTIPYRETIC AND ANALGESIC AGENTS; INHIBITS HORMONE INDUCED UTERINE CONTRACTION; ANTICANCER PROPERTIES; SIDE EFFECT REDUCTION MERCK FROSST CANADA & CO. (CA) 2001-04-24 US disclosed
WO-1996019469-A1 DIARYL-2-(5H)-FURANONES AS COX-2 INHIBITORS MERCK FROSST CANADA INC. (CA) 1996-06-27 WO disclosed