SCHEMBL6995272

SCHEMBL6995272

CCOc1ccc2c(Nc3ccc(Sc4nc(C)cc(C)n4)c(Cl)c3)c(C#N)cnc2c1[N+](=O)[O-]

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 1/20 0.50
EGFR P00533 6/20 0.46
ERBB2 P04626 4/20 0.46
STK4 Q13043 5/20 0.45
IGF1R P08069 7/20 0.42
STK3 Q13188 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7000625 0.88 MAP2K1 (0.53) MAP2K1EGFRERBB2STK4IGF1R
SCHEMBL2203293 0.87 MAP2K1 (0.59) MAP2K1EGFRERBB2STK4IGF1R
SCHEMBL6992049 0.82 IGF1R (0.51) MAP2K1EGFRERBB2IGF1R
SCHEMBL6999694 0.81 MAP2K1 (0.52) MAP2K1EGFRERBB2STK4IGF1R
SCHEMBL2203540 0.81 MAP2K1 (0.58) MAP2K1EGFRERBB2STK4IGF1R
SCHEMBL6998421 0.80 EGFR (0.56) MAP2K1EGFRERBB2STK4STK3
SCHEMBL2203726 0.80 MAP2K1 (0.63) MAP2K1EGFRERBB2STK4IGF1R
SCHEMBL6998072 0.78 MAP2K1 (0.57) MAP2K1EGFRERBB2IGF1R
SCHEMBL7001957 0.77 IGF1R (0.71) MAP2K1EGFRERBB2IGF1R
SCHEMBL6996969 0.77 EGFR (0.57) MAP2K1EGFRERBB2STK4STK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1117659-B1 SUBSTITUTED 3-CYANOQUINOLINES AS PROTEIN TYROSINE KINASES INHIBITORS WYETH CORP (US) 2003-12-03 EP claimed