SCHEMBL6995879

SCHEMBL6995879

Cn1ccc2c1C(=O)N(CCCN1CCN(c3ccc(F)cc3)CC1)CCC2=O

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.48
LMNA P02545 1/20 0.48
MAPK1 P28482 1/20 0.48
DRD3 P35462 6/20 0.48
DRD2 P14416 3/20 0.46
GRIN1 Q05586 1/20 0.43
GRIN2B Q13224 1/20 0.43
DRD4 P21917 2/20 0.42
HTR1A P08908 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6619452 0.92 DRD3 (0.50) KDM4ELMNAMAPK1DRD3DRD2
SCHEMBL6779855 0.89 DRD3 (0.50) KDM4ELMNAMAPK1DRD3DRD2
SCHEMBL6994421 0.89 HTR1A (0.53) DRD3DRD2DRD4HTR1A
SCHEMBL6993564 0.89 KDM4E (0.46) KDM4ELMNAMAPK1DRD3DRD2
SCHEMBL6988326 0.88 DRD3 (0.64) DRD3DRD2DRD4HTR1A
SCHEMBL6989852 0.87 KDM4E (0.47) KDM4ELMNAMAPK1DRD3DRD2
SCHEMBL6989849 0.87 KDM4E (0.47) KDM4ELMNAMAPK1DRD3DRD2
SCHEMBL6990341 0.87 DRD3 (0.54) DRD3DRD2DRD4HTR1A
SCHEMBL6780422 0.85 DRD2 (0.48) KDM4ELMNAMAPK1DRD3DRD2
SCHEMBL6780627 0.85 DRD3 (0.48) KDM4ELMNAMAPK1DRD3DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0557526-B1 PYRROLOAZEPINE COMPOUND SUNTORY LTD (JP) 2003-04-02 EP disclosed
US-5399557-A Cardiovascular disorders SUNTORY LIMITED (JP) 1995-03-21 US disclosed