SCHEMBL6995897

SCHEMBL6995897

CN(CC(COc1ccc(C#N)cc1)N1CC2CC(CN(CCC#N)C2)C1)C(N)=O

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
KCNH2 Q12809 2/20 0.36
HRH3 Q9Y5N1 4/20 0.34
MMP2 P08253 3/20 0.34
HRH2 P25021 2/20 0.34
HRH1 P35367 2/20 0.34
MMP3 P08254 1/20 0.33
GRIN1 Q05586 2/20 0.33
GRIN2B Q13224 2/20 0.33
KCNA5 P22460 2/20 0.33
KDM1A O60341 1/20 0.33
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
JAK3 P52333 1/20 0.33
ABCB11 O95342 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6994726 0.86 HRH2 (0.41) HRH3HRH2HRH1KCNA5
SCHEMBL6995893 0.82 KCNH2 (0.40) ALDH1A1HPGDKCNH2HRH3MMP2
SCHEMBL6990336 0.71 HRH2 (0.35) KCNH2HRH3MMP2HRH2HRH1
SCHEMBL6990334 0.70 HRH2 (0.38) KCNH2HRH3MMP2HRH2HRH1
SCHEMBL6992363 0.70 KCNH2 (0.40) KCNH2HRH3MMP2HRH2HRH1
SCHEMBL6994724 0.68 HRH2 (0.42) KCNH2HRH3HRH2HRH1KCNA5
SCHEMBL6740410 0.68 KCNH2 (0.49) ALDH1A1HPGDKCNH2KDM1A
SCHEMBL6740244 0.67 KCNH2 (0.52) ALDH1A1HPGDKCNH2KDM1A
SCHEMBL6987304 0.67 MCHR1 (0.46) KCNH2HRH3MMP2
SCHEMBL6742821 0.67 KDM4E (0.51) ALDH1A1HPGDKCNH2GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1301510-A1 NEW BISPIDINE COMPOUNDS AND THEIR USE IN THE TREATMENT OF CARDIAC ARRHYTHMIAS AstraZeneca AB (SE) 2003-04-16 EP disclosed
WO-2002004446-A1 NEW BISPIDINE COMPOUNDS AND THEIR USE IN THE TREATMENT OF CARDIAC ARRHYTHMIAS ASTRAZENECA AB (SE) 2002-01-17 WO disclosed