SCHEMBL6995958

SCHEMBL6995958

CC1(C)OC(c2ccc(S(N)(=O)=O)cc2)=C(c2ccc3ccccc3c2)C1=O

nearest known ligand 0.69

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA2 P00918 10/20 0.56
CA1 P00915 8/20 0.56
CA9 Q16790 8/20 0.56
PTGS2 P35354 5/20 0.49
PTGS1 P23219 1/20 0.49
LMNA P02545 1/20 0.47
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
MAPT P10636 1/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
DKK1 O94907 1/20 0.41
GSK3B P49841 1/20 0.41
CA12 O43570 2/20 0.40
PDPK1 O15530 1/20 0.40
CA7 P43166 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6994485 0.89 PTGS2 (0.62) PTGS2PTGS1
SCHEMBL7002002 0.86 PTGS2 (0.56) CA2CA1CA9PTGS2PTGS1
SCHEMBL6999323 0.85 CA2 (0.54) CA2CA1CA9PTGS2PTGS1
SCHEMBL6999849 0.84 CA2 (0.53) CA2CA1CA9PTGS2PTGS1
SCHEMBL6999644 0.84 PTGS2 (0.49) CA2CA1CA9PTGS2PTGS1
SCHEMBL7001251 0.83 CA2 (0.56) CA2CA1CA9PTGS2PTGS1
SCHEMBL7002045 0.82 CA9 (0.52) CA2CA1CA9PTGS2CA12
SCHEMBL6996285 0.82 CA2 (0.42) CA2CA1CA9PTGS2PTGS1
Polmacoxib SCHEMBL3233093 0.82 PTGS2 (0.55) CA2CA1CA9PTGS2PTGS1
Polmacoxib SCHEMBL29351757 0.82 PTGS2 (0.55) CA2CA1CA9PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1109799-B1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORP (KR) 2003-12-17 EP claimed
US-6492416-B1 TREATING INFLAMMATION AND ASSOCIATED DISORDERS PACIFIC CORPORATION (KR) 2002-12-10 US claimed
EP-1109799-B1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORP (KR) 2003-12-17 EP disclosed
US-6492416-B1 TREATING INFLAMMATION AND ASSOCIATED DISORDERS PACIFIC CORPORATION (KR) 2002-12-10 US disclosed