SCHEMBL6997265

SCHEMBL6997265

CC1=C(N)Nc2cc(CNCc3cccc(C)c3C)ccc2O1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
PARP1 P09874 3/20 0.38
HTT P42858 2/20 0.34
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
TP53 P04637 1/20 0.32
MAPK1 P28482 1/20 0.32
MC5R P33032 1/20 0.32
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA9 Q16790 1/20 0.31
DRD4 P21917 1/20 0.31
DRD3 P35462 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6995114 0.99 MEN1 (0.39) MEN1KMT2APARP1HTTALDH1A1
SCHEMBL7002617 0.84 PARP1 (0.41) MEN1KMT2APARP1ALDH1A1MAPK1
Hydrochloric Acid SCHEMBL6998857 0.83 MEN1 (0.44) MEN1KMT2APARP1HTTALDH1A1
Hydrochloric Acid SCHEMBL6995038 0.83 PARP1 (0.40) MEN1KMT2APARP1ALDH1A1MAPK1
Hydrochloric Acid SCHEMBL7713373 0.82 PARP1 (0.53) MEN1KMT2APARP1HTTALDH1A1
Hydrochloric Acid SCHEMBL6310054 0.82 PARP1 (0.42) MEN1KMT2APARP1
SCHEMBL7002250 0.81 PARP1 (0.42) PARP1MAPK1L3MBTL1
SCHEMBL7002470 0.81 PARP1 (0.42) PARP1
Hydrochloric Acid SCHEMBL7000763 0.81 PARP1 (0.43) MEN1KMT2APARP1HTTALDH1A1
Hydrochloric Acid SCHEMBL6999676 0.81 PARP1 (0.43) MEN1KMT2APARP1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015437-B1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN PHARMACEUTICALS SCHERING AG (DE) 2003-12-03 EP claimed