SCHEMBL7002617

SCHEMBL7002617

CC1=C(N)Nc2cc(CNCc3ccccc3F)ccc2O1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.41
PDGFRB P09619 1/20 0.39
KDR P35968 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
MAPK1 P28482 1/20 0.35
THRB P10828 1/20 0.35
ALDH1A1 P00352 1/20 0.35
SCN8A Q9UQD0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6995038 0.99 PARP1 (0.40) PARP1PDGFRBKDRMEN1KMT2A
Hydrochloric Acid SCHEMBL8133176 0.95 PARP1 (0.40) PARP1PDGFRBKDRMEN1KMT2A
Hydrochloric Acid SCHEMBL6998857 0.85 MEN1 (0.44) PARP1MEN1KMT2AMAPK1ALDH1A1
SCHEMBL6994032 0.84 LMNA (0.42) PARP1PDGFRBKDRMEN1KMT2A
Hydrochloric Acid SCHEMBL7713373 0.84 PARP1 (0.53) PARP1PDGFRBKDRMEN1KMT2A
SCHEMBL6997265 0.84 MEN1 (0.40) PARP1MEN1KMT2ACA1CA2
SCHEMBL7002250 0.84 PARP1 (0.42) PARP1PDGFRBKDRMAPK1SCN8A
Hydrochloric Acid SCHEMBL6996205 0.83 PARP1 (0.41) PARP1PDGFRBKDRMEN1KMT2A
Hydrochloric Acid SCHEMBL6995114 0.83 MEN1 (0.39) PARP1MEN1KMT2ACA1CA2
Hydrochloric Acid SCHEMBL7001196 0.83 PARP1 (0.41) PARP1PDGFRBKDRSCN8A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015437-B1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN PHARMACEUTICALS SCHERING AG (DE) 2003-12-03 EP claimed