SCHEMBL6997570

SCHEMBL6997570

CN1C(=O)C2=C(C1=O)c1c([nH]c3ccccc13)Cc1[nH]c3ccccc3c12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 1/20 0.49
SIRT1 Q96EB6 1/20 0.49
ADORA3 P0DMS8 1/20 0.46
ADORA2A P29274 1/20 0.46
ADORA2B P29275 1/20 0.46
ADORA1 P30542 1/20 0.46
ROCK2 O75116 1/20 0.43
GSK3B P49841 1/20 0.42
KDM4E B2RXH2 4/20 0.41
CHRNA7 P36544 1/20 0.41
DRD2 P14416 2/20 0.40
DRD1 P21728 2/20 0.40
DRD4 P21917 2/20 0.40
DRD5 P21918 2/20 0.40
DRD3 P35462 2/20 0.40
CYP1A2 P05177 2/20 0.40
MEN1 O00255 1/20 0.40
GMNN O75496 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7198661 0.81 GSK3B (0.58) SIRT2SIRT1ADORA3ADORA2AADORA2B
SCHEMBL6867398 0.79 CDK4 (0.49) SIRT2GSK3BKDM4EMEN1KMT2A
SCHEMBL6997136 0.78 MPO (0.45) GSK3BDRD2DRD4DRD3ADRA1A
SCHEMBL6995402 0.77 KDM4E (0.41) SIRT2SIRT1ADORA3ADORA2AADORA2B
SCHEMBL7001531 0.77 KDM4E (0.47) SIRT2SIRT1ADORA3ADORA2AADORA2B
SCHEMBL7001489 0.76 SMN1; SMN2 (0.45) SIRT2SIRT1ADORA3ADORA2AADORA2B
SCHEMBL6866221 0.76 SMN1; SMN2 (0.45) SIRT2SIRT1ADORA3ADORA2AADORA2B
SCHEMBL15797027 0.75 GSK3B (0.53) SIRT2SIRT1ADORA3ADORA2AADORA2B
SCHEMBL15797189 0.75 GSK3B (0.53) SIRT2SIRT1ADORA3ADORA2AADORA2B
SCHEMBL6864424 0.74 NQO1 (0.41) SIRT2KDM4EMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1109785-B1 INDOLE DERIVATIVES AND THEIR USE IN THE TREATMENT OF MALIGNANT AND OTHER DISEASES CAUSED BY PATHOLOGICAL CELL PROLIFERATION ZENTARIS AG (DE) 2003-01-02 EP disclosed