SCHEMBL6998028

SCHEMBL6998028

O=C1NCCC(=O)c2c1ccn2CCCCN1CCC(c2nsc3cc(F)ccc23)CC1

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 6/20 0.46
HTR1D P28221 1/20 0.45
HTR1B P28222 1/20 0.45
HTR2A P28223 3/20 0.39
HTR1A P08908 2/20 0.39
HTR6 P50406 1/20 0.38
HTR2C P28335 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7000043 0.87 DRD2 (0.46) DRD2HTR1DHTR1BHTR2AHTR1A
SCHEMBL6993800 0.85 DRD2 (0.47) DRD2HTR1DHTR1BHTR2AHTR1A
SCHEMBL6997100 0.84 DRD2 (0.65) DRD2HTR2AHTR1AHTR6
SCHEMBL6993415 0.74 HTR2A (0.52) DRD2HTR2AHTR6HTR2C
SCHEMBL6997109 0.72 DRD2 (0.46) DRD2HTR2AHTR1AHTR6
SCHEMBL6186847 0.72 HTR1D (0.54) DRD2HTR1DHTR1BHTR2AHTR1A
SCHEMBL1545312 0.71 HTR1D (0.50) DRD2HTR1DHTR1BHTR2AHTR1A
SCHEMBL9117307 0.71 HTR1D (0.50) DRD2HTR1DHTR1BHTR2AHTR1A
Hydrochloric Acid SCHEMBL1545002 0.71 HTR1D (0.49) DRD2HTR1DHTR1BHTR2AHTR1A
SCHEMBL7001825 0.70 DRD2 (0.65) DRD2HTR2AHTR1AHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0915881-B1 PYRROLOAZEPINE COMPOUNDS SUNTORY LTD (JP) 2003-01-08 EP disclosed
US-6211362-B1 CHEMICAL INTERMEDIATE FOR DRUGS SUNTORY LIMITED (JP) 2001-04-03 US disclosed
US-6187772-B1 Pyrroloazepine compounds SUNTORY LIMITED (JP) 2001-02-13 US disclosed