SCHEMBL6997100

SCHEMBL6997100

O=C1NCCC(=O)c2c1ccn2CCCCN1CCC(c2noc3cc(F)ccc23)CC1

nearest known ligand 0.65

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 7/20 0.65
HTR2A P28223 3/20 0.56
ACHE P22303 2/20 0.55
HTR1A P08908 2/20 0.55
SLC6A4 P31645 1/20 0.55
HTR6 P50406 1/20 0.53
KCNH2 Q12809 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7001825 0.87 DRD2 (0.65) DRD2HTR2AACHEHTR1ASLC6A4
SCHEMBL6993106 0.85 DRD2 (0.65) DRD2HTR2AACHEHTR1ASLC6A4
SCHEMBL6998028 0.84 DRD2 (0.46) DRD2HTR2AHTR1AHTR6
SCHEMBL20512946 0.79 DRD2 (1.00) DRD2HTR2AHTR1AHTR6KCNH2
SCHEMBL30179184 0.79 DRD2 (1.00) DRD2HTR2AHTR1AHTR6KCNH2
SCHEMBL8917266 0.78 DRD2 (0.61) DRD2HTR2AACHESLC6A4HTR6
SCHEMBL9995021 0.77 ACHE (0.66) DRD2HTR2AACHEHTR1ASLC6A4
SCHEMBL6780296 0.77 DRD2 (0.61) DRD2HTR2AACHEHTR1ASLC6A4
SCHEMBL1545611 0.76 ACHE (0.93) DRD2HTR2AACHEHTR1ASLC6A4
SCHEMBL9995324 0.76 DRD2 (0.63) DRD2HTR2AACHEHTR1ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0915881-B1 PYRROLOAZEPINE COMPOUNDS SUNTORY LTD (JP) 2003-01-08 EP disclosed
US-6211362-B1 CHEMICAL INTERMEDIATE FOR DRUGS SUNTORY LIMITED (JP) 2001-04-03 US disclosed
US-6187772-B1 Pyrroloazepine compounds SUNTORY LIMITED (JP) 2001-02-13 US disclosed