SCHEMBL6998403

SCHEMBL6998403

COc1ccc2c(c1OC)C[C@H](C1CCN(CCCc3ccccc3)CC1)O[C@@H]2CN

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.46
SIGMAR1 Q99720 3/20 0.45
EBP Q15125 2/20 0.45
TMEM97 Q5BJF2 1/20 0.45
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
EBPL Q9BY08 1/20 0.43
OPRM1 P35372 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6998399 1.00 ABCB1 (0.46) ABCB1SIGMAR1EBPTMEM97KDM4E
SCHEMBL6998407 1.00 ABCB1 (0.46) ABCB1SIGMAR1EBPTMEM97KDM4E
SCHEMBL6999326 0.95 HTR1A (0.43) SIGMAR1EBPTMEM97ALDH1A1
SCHEMBL6999331 0.95 HTR1A (0.43) SIGMAR1EBPTMEM97ALDH1A1
SCHEMBL6999335 0.95 HTR1A (0.43) SIGMAR1EBPTMEM97ALDH1A1
SCHEMBL6995341 0.89 ACHE (0.48) SIGMAR1
SCHEMBL6995337 0.89 ACHE (0.48) SIGMAR1
SCHEMBL6995343 0.89 ACHE (0.48) SIGMAR1
SCHEMBL7001096 0.86 HTR2A (0.49) TMEM97
SCHEMBL6998747 0.85 DRD1 (0.43) SIGMAR1EBPTMEM97ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015446-B1 (4-PIPERIDINYL)-1H-2-BENZOPYRAN DERIVATIVES USEFUL AS ANTIPSYCHOTIC AGENTS AVENTIS PHARMA INC (US) 2003-04-02 EP disclosed
US-6004982-A SIDE EFFECT REDUCTION; SCHIZOPHRENIA HOECHST MARION ROUSSEL, INC. (US) 1999-12-21 US disclosed