SCHEMBL7000628

SCHEMBL7000628

CC1=C(N)Nc2cc(CNCc3ccc(S(C)(=O)=O)cc3)ccc2O1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.41
PTGS2 P35354 4/20 0.35
GHSR Q92847 1/20 0.35
CA1 P00915 5/20 0.35
CA2 P00918 5/20 0.35
CA12 O43570 2/20 0.34
CA9 Q16790 2/20 0.34
PDE5A O76074 1/20 0.34
KMT2A Q03164 1/20 0.34
LMNA P02545 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CNR1 P21554 1/20 0.33
ABL1 P00519 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6990243 0.99 PARP1 (0.41) PARP1PTGS2GHSRCA1CA2
SCHEMBL6999572 0.91 CA1 (0.46) PARP1CA1CA2CA12CA9
Hydrochloric Acid SCHEMBL6993188 0.90 CA1 (0.48) PARP1CA1CA2CA12CA9
Hydrochloric Acid SCHEMBL6999676 0.84 PARP1 (0.43) PARP1KMT2ASMN1; SMN2
Hydrochloric Acid SCHEMBL7000763 0.84 PARP1 (0.43) PARP1CA1CA2CA12CA9
SCHEMBL6994032 0.83 LMNA (0.42) PARP1KMT2ALMNASMN1; SMN2
SCHEMBL6993345 0.83 PARP1 (0.42) PARP1KMT2ALMNASMN1; SMN2
Hydrochloric Acid SCHEMBL7713373 0.83 PARP1 (0.53) PARP1CA1CA2KMT2ASMN1; SMN2
Hydrochloric Acid SCHEMBL6310054 0.83 PARP1 (0.42) PARP1KMT2A
SCHEMBL6995764 0.83 CHRM2 (0.41) PARP1CA1CA2CA12KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015437-B1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN PHARMACEUTICALS SCHERING AG (DE) 2003-12-03 EP claimed