SCHEMBL7001027

SCHEMBL7001027

CCCCCCCC(=O)Nc1nc[nH]c1C#N

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 3/20 0.62
DEGS1 O15121 1/20 0.45
SPHK2 Q9NRA0 1/20 0.44
SPHK1 Q9NYA1 1/20 0.44
RAB9A P51151 2/20 0.44
ALDH1A1 P00352 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
LMNA P02545 2/20 0.43
HPGD P15428 1/20 0.43
TSHR P16473 1/20 0.43
NPC1 O15118 2/20 0.42
GLA P06280 1/20 0.42
MAPK1 P28482 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
POLB P06746 1/20 0.42
CETP P11597 1/20 0.40
GSK3B P49841 1/20 0.40
MAPK8 P45983 1/20 0.40
MAPK9 P45984 1/20 0.40
SOAT1 P35610 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6996417 1.00 XDH (0.62) XDHDEGS1SPHK2SPHK1RAB9A
SCHEMBL6999626 1.00 XDH (0.62) XDHDEGS1SPHK2SPHK1RAB9A
SCHEMBL6996532 0.99 XDH (0.64) XDHDEGS1SPHK2SPHK1RAB9A
SCHEMBL10821714 0.94 XDH (0.58) XDHDEGS1RAB9AALDH1A1SMN1; SMN2
SCHEMBL6999635 0.89 XDH (0.50) XDHALDH1A1GSK3B
SCHEMBL6999473 0.76 SPHK2 (0.47) XDHDEGS1SPHK2SPHK1RAB9A
SCHEMBL7827505 0.75 XDH (0.45) XDHDEGS1SPHK2SPHK1RAB9A
SCHEMBL7052321 0.75 XDH (0.61) XDHDEGS1SPHK2SPHK1RAB9A
SCHEMBL5193809 0.75 XDH (0.61) XDHDEGS1SPHK2SPHK1RAB9A
SCHEMBL6334335 0.75 GABRR1 (0.36) XDHALDH1A1SMN1; SMN2L3MBTL1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1069126-B1 TRIAZOLOPURINE DERIVATIVES, MEDICINAL COMPOSITION CONTAINING THE DERIVATIVES, ADENOSINE A3 RECEPTOR COMPATIBILIZING AGENT, AND ASTHMATIC REMEDY OTSUKA PHARMA CO LTD (JP) 2003-05-28 EP disclosed
US-6288070-B1 Triazolopurine derivatives, medicinal composition containing the derivatives, adenosine A3 receptor compatibilizing agent, and asthmatic remedy OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 2001-09-11 US disclosed