SCHEMBL7827505

SCHEMBL7827505

CCCCCCC(=O)Nc1ncn(C)c1C#N

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.45
DEGS1 O15121 1/20 0.44
RAB9A P51151 2/20 0.43
LMNA P02545 3/20 0.42
ALDH1A1 P00352 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
HPGD P15428 1/20 0.42
TSHR P16473 1/20 0.42
NPC1 O15118 2/20 0.41
GLA P06280 1/20 0.41
MAPK1 P28482 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
POLB P06746 1/20 0.41
KMT2A Q03164 1/20 0.41
SPHK2 Q9NRA0 1/20 0.41
SPHK1 Q9NYA1 1/20 0.41
SOAT1 P35610 4/20 0.40
SOAT2 O75908 2/20 0.40
CETP P11597 1/20 0.39
MAPK8 P45983 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6998288 0.86 XDH (0.44) XDHDEGS1RAB9ALMNAALDH1A1
SCHEMBL7005257 0.82 DEGS1 (0.47) XDHDEGS1RAB9ALMNAALDH1A1
SCHEMBL7003410 0.79 HDAC1 (0.48) TSHRPOLBKMT2ASPHK2SPHK1
SCHEMBL6999626 0.75 XDH (0.62) XDHDEGS1RAB9ALMNAALDH1A1
SCHEMBL7001027 0.75 XDH (0.62) XDHDEGS1RAB9ALMNAALDH1A1
SCHEMBL6996417 0.75 XDH (0.62) XDHDEGS1RAB9ALMNAALDH1A1
SCHEMBL15457577 0.73 EGLN1 (0.44) XDHDEGS1RAB9ALMNAHPGD
SCHEMBL6996532 0.73 XDH (0.64) XDHDEGS1RAB9ALMNAALDH1A1
SCHEMBL7006926 0.73 DEGS1 (0.46) XDHDEGS1RAB9ALMNAALDH1A1
SCHEMBL1573799 0.73 ALDH1A1 (0.41) DEGS1RAB9ALMNAALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6288070-B1 Triazolopurine derivatives, medicinal composition containing the derivatives, adenosine A3 receptor compatibilizing agent, and asthmatic remedy OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 2001-09-11 US disclosed
EP-1069126-A1 TRIAZOLOPURINE DERIVATIVES, MEDICINAL COMPOSITION CONTAINING THE DERIVATIVES, ADENOSINE A3 RECEPTOR COMPATIBILIZING AGENT, AND ASTHMATIC REMEDY OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 2001-01-17 EP disclosed