SCHEMBL7001472

SCHEMBL7001472

CC(C)(C)OC(=O)N1c2c(cccc2C(N)=O)CCC1CO[Si](C)(C)C(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 12/20 0.38
HSD11B1 P28845 1/20 0.35
HTR1A P08908 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7004166 0.91 HSD11B1 (0.35) PARP1HSD11B1
SCHEMBL7001564 0.89 HTR1A (0.35) PARP1HTR1A
SCHEMBL7007832 0.82 MTNR1A (0.38)
SCHEMBL958204 0.76 CHRM2 (0.35) PARP1
SCHEMBL625416 0.76 CHRM2 (0.35) PARP1
SCHEMBL211419 0.76 CHRM2 (0.35) PARP1
SCHEMBL7005115 0.72 ACE (0.41)
SCHEMBL30681463 0.71 SCN9A (0.40)
SCHEMBL30681436 0.71 SCN9A (0.40)
SCHEMBL30681288 0.69 NOTUM (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030105118-A1 Tricyclic quinazolinediones SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2003-06-05 US disclosed
EP-1288216-A1 TRICYCLIC QUINAZOLINEDIONES SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2003-03-05 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030105118-A1 Tricyclic quinazolinediones PARP1, PARP11, PARP2 PARP1 1/4885HSD11B1 1000/4885HTR1A 135/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.