SCHEMBL700153

SCHEMBL700153

CCCCOC(=O)C1NCCc2ccccc21

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.55
NPSR1 Q6W5P4 1/20 0.55
SLC6A2 P23975 1/20 0.44
SLC6A4 P31645 1/20 0.44
OPRM1 P35372 8/20 0.43
OPRK1 P41145 2/20 0.43
SLC18A2 Q05940 1/20 0.43
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
GID4 Q8IVV7 1/20 0.42
PRCP P42785 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
MEN1 O00255 1/20 0.41
MAPT P10636 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9525353 0.87 TSHR (0.55) TSHRNPSR1SLC6A2SLC6A4OPRM1
SCHEMBL23119015 0.87 TSHR (0.60) TSHRNPSR1SLC6A2SLC6A4OPRM1
SCHEMBL4853532 0.87 TSHR (0.60) TSHRNPSR1SLC6A2SLC6A4OPRM1
SCHEMBL9852994 0.86 TSHR (0.57) TSHRNPSR1SLC6A2SLC6A4OPRM1
Hydrochloric Acid SCHEMBL19953531 0.85 TSHR (0.62) TSHRNPSR1SLC6A2SLC6A4OPRM1
Hydrochloric Acid SCHEMBL2790413 0.85 TSHR (0.62) TSHRNPSR1SLC6A2SLC6A4OPRM1
SCHEMBL9526410 0.85 TSHR (0.58) TSHRNPSR1SLC6A2SLC6A4OPRM1
SCHEMBL19398219 0.84 KMT2A (0.39) TSHRNPSR1OPRM1OPRK1SLC18A2
SCHEMBL9853004 0.83 TSHR (0.59) TSHRNPSR1SLC6A2SLC6A4OPRM1
SCHEMBL698946 0.83 TSHR (0.36) TSHRNPSR1SLC18A2TDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421824-A1 AZETIDINYL DIAMIDES AS MONOACYLGLYCEROL LIPASE INHIBITORS Janssen Pharmaceutica N.V. (BE) 2012-02-29 EP disclosed
WO-1999018091-A1 NOVEL COMPOUNDS USEFUL AS NEURO-PROTECTIVE AGENTS ELI LILLY AND COMPANY (US) 1999-04-15 WO disclosed