SCHEMBL698946

SCHEMBL698946

CCCCOC(=O)C1NCCc2c[c]ccc21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.36
NPSR1 Q6W5P4 1/20 0.36
PPARG P37231 3/20 0.34
SLC18A2 Q05940 1/20 0.34
L3MBTL1 Q9Y468 3/20 0.33
TDP1 Q9NUW8 1/20 0.33
MAPK1 P28482 2/20 0.32
KDM4E B2RXH2 1/20 0.32
LMNA P02545 2/20 0.32
CYP1A2 P05177 2/20 0.32
CYP2C19 P33261 2/20 0.32
ESR1 P03372 1/20 0.32
CYP2D6 P10635 1/20 0.32
NR1H2 P55055 1/20 0.32
RNASEL Q05823 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
PDE4D Q08499 1/20 0.32
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL700153 0.83 TSHR (0.55) TSHRNPSR1SLC18A2L3MBTL1TDP1
SCHEMBL19398219 0.80 KMT2A (0.39) TSHRNPSR1SLC18A2KMT2ACA1
SCHEMBL4514045 0.74 TSHR (0.44) TSHRNPSR1
SCHEMBL8803919 0.74 L3MBTL1 (0.36) TSHRPPARGL3MBTL1TDP1MAPK1
SCHEMBL8802238 0.74 TSHR (0.35) TSHRNPSR1PPARGL3MBTL1TDP1
Hydrochloric Acid SCHEMBL4514461 0.73 TSHR (0.47) TSHRNPSR1
Hydrochloric Acid SCHEMBL3878664 0.73 TSHR (0.47) TSHRNPSR1
SCHEMBL699685 0.73 SMN1; SMN2 (0.39) LMNASMN1; SMN2KMT2A
SCHEMBL17748955 0.72 GAA (0.34) TSHRPPARGL3MBTL1TDP1MAPK1
SCHEMBL1967366 0.71 TSHR (0.41) TSHRNPSR1PPARGL3MBTL1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421824-A1 AZETIDINYL DIAMIDES AS MONOACYLGLYCEROL LIPASE INHIBITORS Janssen Pharmaceutica N.V. (BE) 2012-02-29 EP claimed