SCHEMBL7001601

SCHEMBL7001601

COc1cncc(N2C[C@@H]3C[C@H]2CN3C(=O)OC(C)(C)C)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 2/20 0.52
CHRNB2 P17787 5/20 0.49
CHRNA4 P43681 5/20 0.49
HDAC1 Q13547 2/20 0.46
PARP1 P09874 1/20 0.46
HSD11B1 P28845 1/20 0.44
RET P07949 2/20 0.44
CHRNB4 P30926 4/20 0.42
CHRNA3 P32297 4/20 0.42
FGFR1 P11362 1/20 0.41
FGFR2 P21802 1/20 0.41
FGFR4 P22455 1/20 0.41
FGFR3 P22607 1/20 0.41
KDR P35968 1/20 0.41
F13A1 P00488 1/20 0.39
TGM2 P21980 1/20 0.39
TGM1 P22735 1/20 0.39
MAPK8 P45983 1/20 0.39
IDH1 O75874 1/20 0.38
SPR P35270 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2958457 0.93 GPR119 (0.48) GPR119CHRNB2CHRNA4HDAC1PARP1
SCHEMBL2955018 0.90 GPR119 (0.46) GPR119CHRNB2CHRNA4HDAC1PARP1
SCHEMBL2949364 0.86 GPR119 (0.48) GPR119CHRNB2CHRNA4HDAC1PARP1
SCHEMBL11963191 0.86 GPR119 (0.48) GPR119CHRNB2CHRNA4HDAC1PARP1
SCHEMBL3050128 0.86 GPR119 (0.47) GPR119HDAC1PARP1HSD11B1RET
SCHEMBL3050124 0.86 GPR119 (0.47) GPR119HDAC1PARP1HSD11B1RET
SCHEMBL23042937 0.85 GPR119 (0.51) GPR119HDAC1PARP1HSD11B1RET
SCHEMBL5036684 0.85 CHRNB2 (0.57) CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL30261886 0.85 GPR119 (0.51) GPR119HDAC1PARP1HSD11B1RET
SCHEMBL7145919 0.83 CHRNB2 (0.52) GPR119CHRNB2CHRNA4HDAC1PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1147112-B1 DIAZABICYCLIC DERIVATIVES AS NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS ABBOTT LAB (US) 2003-10-29 EP disclosed