SCHEMBL7145919

SCHEMBL7145919

CC(C)(C)OC(=O)N1C[C@@H]2C[C@H]1CN2c1cncc(C(N)=O)c1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.52
CHRNA4 P43681 2/20 0.52
HDAC1 Q13547 2/20 0.47
GPR119 Q8TDV5 3/20 0.46
PARP1 P09874 1/20 0.43
HSD11B1 P28845 1/20 0.41
RET P07949 2/20 0.40
MAPK8 P45983 1/20 0.38
SPR P35270 1/20 0.37
F13A1 P00488 1/20 0.37
TGM2 P21980 1/20 0.37
TGM1 P22735 1/20 0.37
NR1H2 P55055 1/20 0.36
NR1H3 Q13133 1/20 0.36
IDH1 O75874 1/20 0.36
GRM2 Q14416 1/20 0.35
PARP14 Q460N5 1/20 0.34
AR P10275 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2960207 0.85 HDAC1 (0.49) CHRNB2CHRNA4HDAC1GPR119PARP1
SCHEMBL2949364 0.85 GPR119 (0.48) CHRNB2CHRNA4HDAC1GPR119PARP1
SCHEMBL11963191 0.85 GPR119 (0.48) CHRNB2CHRNA4HDAC1GPR119PARP1
SCHEMBL7001601 0.83 GPR119 (0.52) CHRNB2CHRNA4HDAC1GPR119PARP1
SCHEMBL5041416 0.83 CHRNB2 (0.62) CHRNB2CHRNA4HDAC1
SCHEMBL5043514 0.83 CHRNB2 (0.62) CHRNB2CHRNA4HDAC1
SCHEMBL2958457 0.79 GPR119 (0.48) CHRNB2CHRNA4HDAC1GPR119PARP1
SCHEMBL3050128 0.79 GPR119 (0.47) HDAC1GPR119PARP1HSD11B1RET
SCHEMBL3050124 0.79 GPR119 (0.47) HDAC1GPR119PARP1HSD11B1RET
SCHEMBL38661622 0.78 GPR119 (0.52) HDAC1GPR119PARP1HSD11B1RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1359152-A2 Diazabicyclic derivatives as nicotinic acetylcholine receptor ligands ABBOTT LABORATORIES (US) 2003-11-05 EP disclosed