SCHEMBL7001767

SCHEMBL7001767

CC1=C(N)Nc2cc(CNC3Cc4ccccc4C3)ccc2O1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.40
OPRD1 P41143 2/20 0.40
OPRK1 P41145 2/20 0.40
GRIN2B Q13224 6/20 0.38
FYN P06241 1/20 0.38
PARP1 P09874 3/20 0.37
HDAC1 Q13547 1/20 0.36
SIGMAR1 Q99720 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
HTT P42858 1/20 0.33
MAOA P21397 2/20 0.33
KDM1A O60341 1/20 0.33
MAOB P27338 1/20 0.33
SMO Q99835 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7003624 0.99 OPRM1 (0.39) OPRM1OPRD1OPRK1GRIN2BFYN
SCHEMBL6991856 0.82 PRMT5 (0.43) PARP1MAOAMAOB
Hydrochloric Acid SCHEMBL6996290 0.81 PRMT5 (0.43) PARP1MAOAMAOB
SCHEMBL7091667 0.80 PRMT5 (0.51)
Hydrochloric Acid SCHEMBL6989619 0.79 PRMT5 (0.50)
Hydrochloric Acid SCHEMBL7713373 0.77 PARP1 (0.53) PARP1HTT
SCHEMBL6992904 0.75 PARP1 (0.66) FYNPARP1HDAC1MAOB
SCHEMBL7000588 0.74 PARP1 (0.37) PARP1
Hydrochloric Acid SCHEMBL7707646 0.74 MEN1 (0.41) PARP1CYP3A4HTT
Hydrochloric Acid SCHEMBL7000763 0.73 PARP1 (0.43) PARP1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015437-B1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN PHARMACEUTICALS SCHERING AG (DE) 2003-12-03 EP claimed