SCHEMBL6991856

SCHEMBL6991856

CC1=C(N)Nc2cc(CNC3CCc4ccccc43)ccc2O1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PRMT5 O14744 1/20 0.43
KDM4E B2RXH2 5/20 0.42
MAOA P21397 3/20 0.41
MAOB P27338 3/20 0.41
HTR6 P50406 2/20 0.41
BCHE P06276 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
ACHE P22303 1/20 0.41
ADRA1A P35348 1/20 0.41
HRH3 Q9Y5N1 1/20 0.39
PDPK1 O15530 1/20 0.38
ALDH1A1 P00352 2/20 0.36
KMT2A Q03164 1/20 0.35
DHFR P00374 1/20 0.35
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
PARP1 P09874 2/20 0.34
MPO P05164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6996290 0.99 PRMT5 (0.43) PRMT5KDM4EMAOAMAOBHTR6
SCHEMBL7091667 0.94 PRMT5 (0.51) PRMT5KDM4EALDH1A1KMT2ADHFR
Hydrochloric Acid SCHEMBL6989619 0.93 PRMT5 (0.50) PRMT5KDM4EALDH1A1KMT2ADHFR
SCHEMBL7001767 0.82 OPRM1 (0.40) MAOAMAOBPARP1
Hydrochloric Acid SCHEMBL7003624 0.81 OPRM1 (0.39) MAOAMAOBKMT2APARP1
SCHEMBL6999674 0.78 PARP1 (0.60) PRMT5KDM4EMAOAMAOBHTR6
Hydrochloric Acid SCHEMBL7713373 0.73 PARP1 (0.53) KDM4EBCHEALDH1A1KMT2ACA1
SCHEMBL6991849 0.73 SIGMAR1 (0.30)
Hydrochloric Acid SCHEMBL6996287 0.72 SIGMAR1 (0.31)
SCHEMBL6988613 0.72 PARP1 (0.58) PRMT5KDM4EALDH1A1KMT2APARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015437-B1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN PHARMACEUTICALS SCHERING AG (DE) 2003-12-03 EP claimed