SCHEMBL7001771

SCHEMBL7001771

CC1Oc2ccc(CNC3Cc4ccccc4C3)cc2N=C1N

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.38
OPRD1 P41143 2/20 0.38
OPRK1 P41145 2/20 0.38
GRIN2B Q13224 6/20 0.38
FYN P06241 1/20 0.38
CTSD P07339 1/20 0.34
PARP1 P09874 1/20 0.34
HDAC1 Q13547 1/20 0.34
SIGMAR1 Q99720 1/20 0.33
KDM1A O60341 2/20 0.33
MAOA P21397 2/20 0.33
MAOB P27338 2/20 0.33
LTA4H P09960 1/20 0.33
DRD2 P14416 1/20 0.32
NR1I3 Q14994 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7003628 0.99 OPRM1 (0.38) OPRM1OPRD1OPRK1GRIN2BFYN
SCHEMBL6991860 0.82 KDM4E (0.42) MAOAMAOBALDH1A1
Hydrochloric Acid SCHEMBL7708035 0.81 KDM4E (0.41) MAOAMAOBALDH1A1NOS3NOS1
SCHEMBL27466929 0.80 PARP1 (0.53) PARP1DRD2ALDH1A1NOS3NOS1
Hydrochloric Acid SCHEMBL6989622 0.79 KDM4E (0.48) ALDH1A1
SCHEMBL6611984 0.79 PARP1 (0.45) PARP1ALDH1A1NOS3NOS1NOS2
Hydrochloric Acid SCHEMBL7713375 0.79 PARP1 (0.52) PARP1DRD2ALDH1A1NOS3NOS1
Hydrochloric Acid SCHEMBL6302797 0.78 PARP1 (0.44) PARP1ALDH1A1NOS3NOS1NOS2
SCHEMBL6610312 0.78 PARP1 (0.51) PARP1ALDH1A1NOS3NOS1NOS2
Hydrochloric Acid SCHEMBL6302705 0.77 NOS1 (0.46) PARP1ALDH1A1NOS3NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015437-B1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN PHARMACEUTICALS SCHERING AG (DE) 2003-12-03 EP claimed