SCHEMBL7001994

SCHEMBL7001994

CN1CCC(O)(c2cccc(Cl)c2)C(C(=O)c2cccc(Cl)c2)C1

nearest known ligand 0.68

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.68
ALDH1A1 P00352 4/20 0.68
MAPT P10636 3/20 0.68
SLC6A3 Q01959 3/20 0.67
LMNA P02545 3/20 0.65
CNR2 P34972 1/20 0.48
MEN1 O00255 1/20 0.48
MAPK1 P28482 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.45
KDM2B Q8NHM5 4/20 0.44
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7004017 0.81 KMT2A (1.00) KMT2AALDH1A1MAPTSLC6A3LMNA
SCHEMBL4194116 0.80 SLC6A3 (1.00) KMT2AALDH1A1MAPTSLC6A3LMNA
SCHEMBL6997233 0.79 KMT2A (1.00) KMT2AALDH1A1MAPTSLC6A3LMNA
SCHEMBL7002087 0.78 SLC6A3 (0.79) KMT2AALDH1A1MAPTSLC6A3LMNA
SCHEMBL7001626 0.78 KMT2A (0.70) KMT2AALDH1A1MAPTSLC6A3LMNA
SCHEMBL6995030 0.76 SLC6A3 (0.69) KMT2AALDH1A1MAPTSLC6A3LMNA
SCHEMBL7001985 0.73 KMT2A (0.79) KMT2AALDH1A1MAPTSLC6A3LMNA
SCHEMBL10849364 0.72 SLC6A3 (0.42) KMT2AALDH1A1MAPTSLC6A3LMNA
SCHEMBL10655679 0.72 SLC6A3 (0.42) KMT2AALDH1A1MAPTSLC6A3LMNA
SCHEMBL10655688 0.72 SLC6A3 (0.42) KMT2AALDH1A1MAPTSLC6A3LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242080-A4 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE UNIV GEORGETOWN (US) 2003-01-22 EP claimed
EP-1242080-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2002-09-25 EP claimed
WO-2001022964-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2001-04-05 WO claimed
EP-1242080-A4 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE UNIV GEORGETOWN (US) 2003-01-22 EP disclosed
EP-1242080-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2002-09-25 EP disclosed
WO-2001022964-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2001-04-05 WO disclosed