SCHEMBL7002087

SCHEMBL7002087

Cc1cc(C(=O)C2CN(C)CCC2(O)c2ccc(Cl)c(C)c2)ccc1Cl

nearest known ligand 0.79

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 6/20 0.79
KMT2A Q03164 6/20 0.67
ALDH1A1 P00352 4/20 0.67
MAPT P10636 3/20 0.67
LMNA P02545 3/20 0.67
MEN1 O00255 1/20 0.40
MAPK1 P28482 1/20 0.40
OPRM1 P35372 1/20 0.38
CCR2 P41597 1/20 0.36
KDM2B Q8NHM5 1/20 0.35
AR P10275 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6995030 0.90 SLC6A3 (0.69) SLC6A3KMT2AALDH1A1MAPTLMNA
SCHEMBL4194116 0.88 SLC6A3 (1.00) SLC6A3KMT2AALDH1A1MAPTLMNA
SCHEMBL6997233 0.81 KMT2A (1.00) SLC6A3KMT2AALDH1A1MAPTLMNA
SCHEMBL7001985 0.79 KMT2A (0.79) SLC6A3KMT2AALDH1A1MAPTLMNA
SCHEMBL7001626 0.79 KMT2A (0.70) SLC6A3KMT2AALDH1A1MAPTLMNA
SCHEMBL7001403 0.78 SLC6A3 (0.78) SLC6A3KMT2AALDH1A1MAPTLMNA
SCHEMBL7001994 0.78 KMT2A (0.68) SLC6A3KMT2AALDH1A1MAPTLMNA
SCHEMBL7003749 0.76 KMT2A (0.77) SLC6A3KMT2AALDH1A1MAPTLMNA
Flazalone SCHEMBL43716 0.76 KMT2A (1.00) SLC6A3KMT2AALDH1A1MAPTLMNA
SCHEMBL6998081 0.76 KMT2A (0.77) SLC6A3KMT2AALDH1A1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242080-A4 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE UNIV GEORGETOWN (US) 2003-01-22 EP claimed
EP-1242080-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2002-09-25 EP claimed
WO-2001022964-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2001-04-05 WO claimed
EP-1242080-A4 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE UNIV GEORGETOWN (US) 2003-01-22 EP disclosed
EP-1242080-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2002-09-25 EP disclosed
WO-2001022964-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2001-04-05 WO disclosed