SCHEMBL7002103

SCHEMBL7002103

CSc1ccc(C2=C(c3cccc(C(F)(F)F)c3)C(=O)C(C)(C)O2)c(F)c1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 3/20 0.38
AKR1C2 P52895 3/20 0.38
PTGES O14684 1/20 0.35
PTGS1 P23219 1/20 0.35
ABCG2 Q9UNQ0 1/20 0.33
CTSD P07339 1/20 0.33
BACE1 P56817 1/20 0.33
KCNA3 P22001 1/20 0.33
PARP10 Q53GL7 1/20 0.33
PARP11 Q9NR21 1/20 0.33
NOTUM Q6P988 1/20 0.33
PGR P06401 1/20 0.32
BRD4 O60885 1/20 0.32
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6996567 0.87 PTGS2 (0.40) AKR1C3AKR1C2PTGS1PGR
SCHEMBL6997650 0.86 PTGS2 (0.38) PTGS1CTSDBACE1NOTUMPGR
SCHEMBL6995715 0.86 PTGS2 (0.43) AKR1C3AKR1C2PTGS1
SCHEMBL6996397 0.85 GSK3B (0.43) AKR1C3AKR1C2PTGS1PGR
SCHEMBL6997353 0.82 PTGS2 (0.43) AKR1C3AKR1C2PTGS1
SCHEMBL6997443 0.82 AKR1C3 (0.38) AKR1C3AKR1C2PTGESPTGS1CTSD
SCHEMBL6998165 0.82 PTGS2 (0.36) AKR1C3AKR1C2PTGS1PGR
SCHEMBL7000249 0.82 KDM4E (0.39) AKR1C3AKR1C2PTGS1
SCHEMBL6999283 0.81 PTGS2 (0.33) AKR1C3AKR1C2PTGS1PGR
SCHEMBL6997325 0.81 PTGS2 (0.36) AKR1C3AKR1C2PTGS1PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1109799-B1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORP (KR) 2003-12-17 EP claimed
US-6492416-B1 TREATING INFLAMMATION AND ASSOCIATED DISORDERS PACIFIC CORPORATION (KR) 2002-12-10 US claimed
EP-1109799-B1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORP (KR) 2003-12-17 EP disclosed
US-6492416-B1 TREATING INFLAMMATION AND ASSOCIATED DISORDERS PACIFIC CORPORATION (KR) 2002-12-10 US disclosed