SCHEMBL7002153

SCHEMBL7002153

CC1=C(N)Nc2cc(C(N)C(=O)OC(C)(C)CCc3cccc(C(F)(F)F)c3)ccc2O1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.35
GRM3 Q14832 1/20 0.35
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
EPHX1 P07099 6/20 0.33
KDM4E B2RXH2 3/20 0.33
ALOX5 P09917 1/20 0.33
FFAR4 Q5NUL3 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
TAAR1 Q96RJ0 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
THRB P10828 1/20 0.32
MC4R P32245 1/20 0.32
ALDH1A1 P00352 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
MMP1 P03956 1/20 0.32
MMP12 P39900 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6994386 0.90 ALOX5 (0.31) KDM4EALOX5
SCHEMBL8137237 0.89 ALOX5 (0.35) ALOX5
SCHEMBL7001571 0.88 GRM2 (0.34) GRM2GRM3ALOX5MEN1KMT2A
SCHEMBL7003205 0.88 GRM2 (0.37) GRM2GRM3KDM4EMEN1KMT2A
SCHEMBL7002397 0.85 ALOX5 (0.31) ALOX5
SCHEMBL6992660 0.85 PDE1C (0.35) MEN1KMT2ATDP1
SCHEMBL6993302 0.85 ALOX5 (0.32) ALOX5
SCHEMBL6994308 0.85 CYP3A4 (0.32) ALOX5
SCHEMBL7001710 0.84 FFAR1 (0.32) SMN1; SMN2
SCHEMBL6997495 0.83 ADRB2 (0.39) MEN1KMT2ATAAR1ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015437-B1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN PHARMACEUTICALS SCHERING AG (DE) 2003-12-03 EP disclosed