SCHEMBL7002218

SCHEMBL7002218

CN(C)C(c1ccc(C#N)cc1)n1c(=O)c2cc(Br)ccc2n2cnnc12.Cc1ccc2c(c1)c(=O)n(Cc1cccnc1)c1nnc(N3CCCCCC3)n21

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.33
GABRA5 P31644 1/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
KDM4E B2RXH2 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
PKM P14618 1/20 0.32
CYP2C19 P33261 1/20 0.32
PIK3R1 P27986 2/20 0.31
PIK3CA P42336 2/20 0.31
ALDH1A1 P00352 1/20 0.31
GLA P06280 1/20 0.31
GAA P10253 1/20 0.31
HPGD P15428 1/20 0.31
CASP1 P29466 1/20 0.31
CASP7 P55210 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7002215 0.84 PIK3R1 (0.36) GABRA1GABRA5MEN1KMT2AKDM4E
SCHEMBL7526734 0.79 PIK3R1 (0.35) PIK3R1PIK3CALMNA
SCHEMBL6854914 0.78 PKM (0.48) GABRA1GABRA5MEN1KMT2AKDM4E
SCHEMBL6854127 0.78 MAPT (0.43) KDM4EALDH1A1HPGDCASP1HSD17B10
SCHEMBL6855211 0.77 PKM (0.49) GABRA1GABRA5MEN1KMT2AKDM4E
SCHEMBL6855386 0.77 MAPT (0.44) KDM4EALDH1A1HPGDCASP1HSD17B10
SCHEMBL7530001 0.77 PDE7A (0.33) PIK3R1PIK3CAALDH1A1LMNATSHR
SCHEMBL6854433 0.76 PIK3R1 (0.36) PIK3R1PIK3CAHSD17B10
SCHEMBL6856311 0.76 SMN1; SMN2 (0.33) HSD17B10
SCHEMBL6994280 0.75 DHFR (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177195-B1 1-AMINO TRIAZOLO 4,3-a! QUINAZOLINE-5-ONES AND OR -5-THIONES INHIBITING PHOSPHODIESTERASE IV WARNER LAMBERT CO (US) 2003-03-19 EP claimed