SCHEMBL7002298

SCHEMBL7002298

CCOC(=O)Oc1c(-c2ccc(SC)cc2)c(-c2ccc(F)cc2)n2c1CCC2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.46
KMT2A Q03164 5/20 0.43
PDE3B Q13370 2/20 0.39
PDE3A Q14432 2/20 0.39
PTGS1 P23219 2/20 0.38
ALDH1A1 P00352 2/20 0.37
LMNA P02545 1/20 0.37
HTT P42858 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
KDM4E B2RXH2 1/20 0.36
MAPK1 P28482 2/20 0.34
GABRG2 P18507 1/20 0.34
GABRB3 P28472 1/20 0.34
GABRA5 P31644 1/20 0.34
GABRA2 P47869 1/20 0.34
GABRB2 P47870 1/20 0.34
MEN1 O00255 2/20 0.33
MAPK14 Q16539 1/20 0.33
GAA P10253 1/20 0.33
OPRM1 P35372 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6995346 0.92 PTGS2 (0.46) PTGS2KMT2APDE3BPDE3APTGS1
SCHEMBL6999021 0.89 KMT2A (0.48) KMT2APDE3BPDE3APTGS1ALDH1A1
SCHEMBL7008536 0.87 RIPK3 (0.45) KMT2APDE3BPDE3AMAPK14
SCHEMBL7012237 0.87 RIPK3 (0.45) KMT2APDE3BPDE3AMAPK14
SCHEMBL6998740 0.86 PTGS2 (0.48) PTGS2KMT2APDE3BPDE3APTGS1
SCHEMBL7006189 0.85 RIPK3 (0.44) KMT2APDE3BPDE3AMAPK14
SCHEMBL6483652 0.84 KMT2A (0.50) PTGS2KMT2APDE3BPDE3APTGS1
SCHEMBL6485382 0.82 KMT2A (0.50) PTGS2KMT2APDE3BPDE3APTGS1
SCHEMBL7006565 0.80 MAPK14 (0.44) KMT2APDE3BPDE3AMAPK14
SCHEMBL7010615 0.80 MAPK14 (0.44) KMT2APDE3BPDE3AMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1246825-B1 FUSED PYRROLE COMPOUNDS, PHARMACEUTICAL AGENTS CONTAINING THE SAME, AND THE USE THEREOF MERCKLE GMBH (DE) 2003-12-17 EP disclosed