SCHEMBL7002884

SCHEMBL7002884

Nc1ccc2[nH]cc(CCCCc3c[nH]c4ccc(N)cc34)c2c1

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.67
CYP2C19 P33261 1/20 0.67
MPO P05164 6/20 0.59
HTR1A P08908 8/20 0.56
HTR1D P28221 8/20 0.56
HTR2A P28223 7/20 0.56
HTR1B P28222 6/20 0.56
TRPM8 Q7Z2W7 4/20 0.56
HTR2C P28335 3/20 0.56
HTR2B P41595 2/20 0.56
CYP1A2 P05177 2/20 0.56
TSHR P16473 2/20 0.56
HTR7 P34969 2/20 0.56
HTR6 P50406 2/20 0.56
HTR4 Q13639 2/20 0.56
HTR3E A5X5Y0 1/20 0.56
HTR3B O95264 1/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2D6 P10635 1/20 0.56
CYP2C9 P11712 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8544422 0.92 HPGD (0.58) HPGDCYP2C19MPOHTR1AHTR1D
SCHEMBL14160299 0.90 HTR1A (0.65) HPGDCYP2C19MPOHTR1AHTR1D
SCHEMBL8978738 0.90 HPGD (0.64) HPGDCYP2C19MPOHTR1AHTR1D
SCHEMBL2847185 0.89 HTR1D (0.70) HPGDCYP2C19MPOHTR1AHTR1D
Hydrochloric Acid SCHEMBL27517910 0.89 HTR1A (0.68) HPGDCYP2C19MPOHTR1AHTR1D
SCHEMBL3379714 0.86 SLC6A4 (0.70) HPGDCYP2C19MPOHTR1AHTR1D
SCHEMBL8235788 0.86 CYP2C19 (0.63) HPGDCYP2C19MPOHTR1AHTR1D
SCHEMBL3878356 0.86 HTR2C (0.68) HPGDCYP2C19MPOHTR1AHTR1D
SCHEMBL27792207 0.85 HPGD (0.58) HPGDCYP2C19MPOHTR1AHTR1D
SCHEMBL9664523 0.83 MPO (0.66) HPGDCYP2C19MPOHTR1AHTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1337511-A1 BIS-HETEROCYCLIC COMPOUNDS WITH ANTITUMOUR AND CHEMOSENSITISING ACTIVITY Sigma-Tau Industrie Farmaceutiche Riunite S.p.A. (IT) 2003-08-27 EP disclosed
WO-2002036561-A1 BIS-HETEROCYCLIC COMPOUNDS WITH ANTITUMOUR AND CHEMOSENSITISING ACTIVITY SIGMA-TAU INDUSTRIE FARMACEUTICHE RIUNITE S.P.A. (IT) 2002-05-10 WO disclosed