SCHEMBL8978738

SCHEMBL8978738

Nc1ccc2[nH]cc(CCCO)c2c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.64
CYP2C19 P33261 1/20 0.64
HTR2C P28335 4/20 0.55
HTR2A P28223 6/20 0.54
HTR1A P08908 3/20 0.54
HTR1D P28221 3/20 0.54
HTR7 P34969 3/20 0.54
HTR2B P41595 2/20 0.54
CYP2D6 P10635 2/20 0.54
CYP1A2 P05177 2/20 0.54
TSHR P16473 2/20 0.54
HTR1B P28222 2/20 0.54
HTR5A P47898 2/20 0.54
HTR6 P50406 2/20 0.54
HTR3E A5X5Y0 1/20 0.54
HTR3B O95264 1/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2C9 P11712 1/20 0.54
DRD1 P21728 1/20 0.54
HTR1E P28566 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3878356 0.90 HTR2C (0.68) HPGDCYP2C19HTR2CHTR2AHTR1A
SCHEMBL7002884 0.90 HPGD (0.67) HPGDCYP2C19HTR2CHTR2AHTR1A
SCHEMBL14160299 0.84 HTR1A (0.65) HPGDCYP2C19HTR2AHTR1AHTR1D
SCHEMBL2847185 0.83 HTR1D (0.70) HPGDCYP2C19HTR2CHTR2AHTR1A
SCHEMBL8544422 0.83 HPGD (0.58) HPGDCYP2C19HTR2CHTR2AHTR1A
Hydrochloric Acid SCHEMBL27517910 0.83 HTR1A (0.68) HPGDCYP2C19HTR2CHTR2AHTR1A
SCHEMBL8630044 0.81 HTR1A (0.56) HTR2CHTR2AHTR1AHTR1DHTR7
SCHEMBL891985 0.81 SLC6A4 (0.67) HTR2CHTR2AHTR1AHTR1DHTR7
SCHEMBL4352009 0.81 MPO (0.74) HTR2AHTR1AMPOSLC6A4TRPM8
SCHEMBL8261013 0.81 SLC6A4 (0.67) HTR2CHTR2AHTR1AHTR1DHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5521188-A Antimigraine cyclobutenedione derivatives of indolylalkyl-pyridinyl and pyrimidinylpiperazines BRISTOL-MYERS SQUIBB COMPANY (US) 1996-05-28 US disclosed
EP-0645385-A1 Antimigraine cyclobutenedione derivatives of indolylalkyl-pyridinyl and pyrimidinylpiperazines Bristol-Myers Squibb Company (US) 1995-03-29 EP disclosed