SCHEMBL7003057

SCHEMBL7003057

CN1CCC(O)(c2ccc(Cl)c(Cl)c2)[CH]C1c1ccc(Cl)c(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 9/20 0.41
OPRM1 P35372 2/20 0.40
SLC6A2 P23975 8/20 0.39
SLC6A4 P31645 8/20 0.39
KCNH2 Q12809 5/20 0.39
CYP2D6 P10635 4/20 0.39
CYP2C19 P33261 3/20 0.39
CYP3A4 P08684 3/20 0.39
CYP1A1 P04798 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2C9 P11712 1/20 0.39
CHRNA1 P02708 1/20 0.39
CHRNG P07510 1/20 0.39
CHRNB1 P11230 1/20 0.39
CHRNB2 P17787 1/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
CHRNA4 P43681 1/20 0.39
CHRND Q07001 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3122638 0.65 OPRM1 (0.52) SLC6A3OPRM1SLC6A2SLC6A4KCNH2
SCHEMBL12497571 0.64 OPRM1 (0.59) SLC6A3OPRM1SLC6A2SLC6A4KCNH2
SCHEMBL11653008 0.64 SLC6A3 (0.46) SLC6A3OPRM1SLC6A2SLC6A4KCNH2
SCHEMBL17186690 0.63 SLC6A4 (0.50) SLC6A3SLC6A2SLC6A4
SCHEMBL14318603 0.63 DRD2 (0.62) SLC6A3OPRM1SLC6A2SLC6A4
SCHEMBL3860327 0.62 DRD2 (0.57) OPRM1
SCHEMBL7001403 0.61 SLC6A3 (0.78) SLC6A3OPRM1SLC6A2SLC6A4KCNH2
SCHEMBL28148678 0.61 ESR2 (0.59) SLC6A3OPRM1SLC6A2SLC6A4KCNH2
SCHEMBL18596508 0.61 SLC6A4 (0.49) SLC6A3SLC6A2SLC6A4KCNH2CYP2D6
SCHEMBL6169426 0.61 SLC6A4 (0.58) SLC6A3OPRM1SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242080-A4 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE UNIV GEORGETOWN (US) 2003-01-22 EP disclosed
EP-1242080-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2002-09-25 EP disclosed
WO-2001022964-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2001-04-05 WO disclosed