SCHEMBL7003987

SCHEMBL7003987

O=C1[N]c2cc(S(=O)(=O)C(F)(F)F)ccc2N1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.44
ESPL1 Q14674 1/20 0.40
POLB P06746 1/20 0.38
MIF P14174 1/20 0.37
PTPRZ1 P23471 1/20 0.36
EPAS1 Q99814 8/20 0.36
LMNA P02545 3/20 0.35
HTT P42858 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
MAPK1 P28482 1/20 0.34
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
PTPN1 P18031 1/20 0.33
KIF11 P52732 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6264592 0.71 CA1 (0.40) KMT2ACYP2C19
SCHEMBL13657421 0.69 GAA (0.56) SMN1; SMN2MEN1KMT2AKIF11
SCHEMBL6221498 0.68 KIF11 (0.40) ALDH1A1MEN1KMT2AKIF11
SCHEMBL1401519 0.67 ROS1 (0.41) ALDH1A1POLBLMNAHTTSMN1; SMN2
SCHEMBL4382993 0.67 TGM2 (0.44) POLBLMNAHTTMEN1KMT2A
SCHEMBL473854 0.67 TGM2 (0.44) MEN1KMT2A
SCHEMBL4752422 0.67 CES1 (0.44) ALDH1A1LMNASMN1; SMN2CYP3A4CYP2D6
SCHEMBL1695075 0.67 CA9 (0.38) ALDH1A1HTTSMN1; SMN2MEN1KMT2A
SCHEMBL4753132 0.67 TGM2 (0.44) MEN1KMT2A
SCHEMBL3817144 0.67 CES1 (0.44) ALDH1A1LMNASMN1; SMN2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347982-A2 SPIRO ISOBENZOFURAN-1,4'-PIPERIDIN]-3-ONES AND 3H-SPIROISOBENZOFURAN-1,4'-PIPERIDINES Neurogen Corporation (US) 2003-10-01 EP disclosed
WO-2002048152-A2 SPIRO[ISOBENZOFURAN-1,4'-PIPERIDIN]-3-ONES AND 3H-SPIROISOBENZOFURAN-1,4'-PIPERIDINES NEUROGEN CORPORATION (US) 2002-06-20 WO disclosed