SCHEMBL7004047

SCHEMBL7004047

OCC1CSc2cccnc2O1

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.34
LTA4H P09960 3/20 0.33
TRPM5 Q9NZQ8 2/20 0.33
NISCH Q9Y2I1 1/20 0.31
HTR2B P41595 1/20 0.31
P2RX7 Q99572 4/20 0.31
CYP1A2 P05177 2/20 0.30
CYP2C19 P33261 2/20 0.30
CYP2C9 P11712 1/20 0.30
ADRA1A P35348 1/20 0.30
TP53 P04637 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
TSHR P16473 1/20 0.30
HIF1A Q16665 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7004199 0.76 LMNA (0.46) LTA4HTP53TSHR
SCHEMBL6097642 0.73 ADRA1A (0.45) NISCHHTR2BCYP1A2CYP2C19ADRA1A
SCHEMBL31343493 0.70 CYP2A6 (0.35) CYP2A6LTA4HNISCHCYP1A2CYP2C19
SCHEMBL4955102 0.70 LTA4H (0.51) LTA4H
SCHEMBL3848567 0.70 LTA4H (0.51) LTA4H
SCHEMBL4955093 0.70 LTA4H (0.51) LTA4H
SCHEMBL4959265 0.67 NISCH (0.35) CYP2A6LTA4HNISCH
SCHEMBL6866771 0.67 CHRNB4 (0.47) LTA4HCYP1A2CYP2C19ADRA1ACYP3A4
SCHEMBL31191058 0.67 CHRNB4 (0.47) LTA4HCYP1A2CYP2C19ADRA1ACYP3A4
SCHEMBL16830889 0.66 CYP2A6 (0.31) CYP2A6LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1296987-A1 COMPOUNDS FOR TREATING IMPAIRED FUNDIC RELAXATION JANSSEN PHARMACEUTICA N.V. (BE) 2003-04-02 EP disclosed
WO-2001098306-A1 COMPOUNDS FOR TREATING IMPAIRED FUNDIC RELAXATION JANSSEN PHARMACEUTICA N.V. (BE) 2001-12-27 WO disclosed