SCHEMBL7006318

SCHEMBL7006318

O=C(O)c1cc(F)c(Br)c(CO)c1F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 2/20 0.37
NFE2L2 Q16236 1/20 0.37
KDM4E B2RXH2 3/20 0.33
ASPH Q12797 2/20 0.33
KDM8 Q8N371 2/20 0.33
PRKAB2 O43741 3/20 0.33
PRKAG1 P54619 3/20 0.33
PRKAA2 P54646 3/20 0.33
PRKAA1 Q13131 3/20 0.33
PRKAG3 Q9UGI9 3/20 0.33
PRKAG2 Q9UGJ0 3/20 0.33
PRKAB1 Q9Y478 3/20 0.33
PTPN1 P18031 1/20 0.33
TSHR P16473 2/20 0.32
AKR1C2 P52895 3/20 0.32
AKR1C1 Q04828 3/20 0.32
AKR1C3 P42330 2/20 0.32
ALB P02768 1/20 0.32
AKR1C4 P17516 1/20 0.32
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL543099 0.79 KEAP1 (0.40) KEAP1NFE2L2KDM4EASPHKDM8
SCHEMBL10515953 0.79 KEAP1 (0.42) KEAP1NFE2L2KDM4EASPHKDM8
SCHEMBL7006447 0.79 KEAP1 (0.38) KEAP1NFE2L2KDM4EASPHKDM8
SCHEMBL7008840 0.78 CA2 (0.42) KEAP1NFE2L2KDM4ETSHRHSD17B10
SCHEMBL19478153 0.77 DRD4 (0.34)
SCHEMBL8056962 0.75 KEAP1 (0.42) KEAP1NFE2L2KDM4EASPHKDM8
SCHEMBL31034649 0.75 KEAP1 (0.42) KEAP1NFE2L2KDM4EASPHKDM8
SCHEMBL23496686 0.74 KEAP1 (0.47) KEAP1NFE2L2KDM4EASPHKDM8
SCHEMBL2670263 0.74 KEAP1 (0.39) KEAP1NFE2L2KDM4EASPHKDM8
SCHEMBL21358502 0.72 AKR1C2 (0.44) KEAP1NFE2L2KDM4EASPHKDM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0775702-B1 NOVEL QUINOLONE- OR NAPHTHYRIDONECARBOXYLIC ACID DERIVATIVE OR SALT THEREOF TOYAMA CHEMICAL CO LTD (JP) 2003-07-23 EP disclosed
US-5935952-A ANTIBACTERIAL AGENT TOYAMA CHEMICAL CO., LTD. (JP) 1999-08-10 US disclosed
EP-0775702-A1 NOVEL QUINOLONE- OR NAPHTHYRIDONECARBOXYLIC ACID DERIVATIVE OR SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 1997-05-28 EP disclosed