SCHEMBL7006728

SCHEMBL7006728

O=C(O)c1cc(Cl)c(F)c(Cl)c1F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.42
NFE2L2 Q16236 1/20 0.42
TSHR P16473 3/20 0.42
ALDH1A1 P00352 3/20 0.42
TP53 P04637 1/20 0.42
CASP1 P29466 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
AKR1C4 P17516 1/20 0.41
AKR1C3 P42330 1/20 0.41
AKR1C2 P52895 1/20 0.41
AKR1C1 Q04828 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
KDM4E B2RXH2 2/20 0.40
MAPT P10636 2/20 0.40
HTT P42858 2/20 0.40
PKM P14618 1/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30255617 0.84 MEN1 (0.37) KEAP1NFE2L2TSHRALDH1A1TP53
SCHEMBL8727193 0.84 ALDH1A1 (0.40) KEAP1NFE2L2TSHRALDH1A1TP53
SCHEMBL5591588 0.84 MEN1 (0.37) KEAP1NFE2L2TSHRALDH1A1TP53
SCHEMBL8683261 0.84 KEAP1 (0.44) KEAP1NFE2L2TSHRALDH1A1TP53
SCHEMBL7005963 0.83 AKR1C2 (0.52) KEAP1NFE2L2TSHRALDH1A1TP53
SCHEMBL29376622 0.83 KEAP1 (0.52) KEAP1NFE2L2TSHRALDH1A1TP53
SCHEMBL8679913 0.83 KEAP1 (0.42) KEAP1NFE2L2TSHRALDH1A1TP53
SCHEMBL2434231 0.83 KEAP1 (0.52) KEAP1NFE2L2TSHRALDH1A1TP53
SCHEMBL23513273 0.82 NOTUM (0.42) KEAP1NFE2L2TSHRALDH1A1TP53
SCHEMBL23496860 0.82 MAP2K1 (0.39) KEAP1NFE2L2TSHRALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0894784-B1 4-FLUOROSALICYLIC ACID DERIVATIVES AND PROCESS FOR PRODUCING THE SAME IHARA CHEMICAL IND CO (JP) 2003-01-08 EP disclosed
US-6166246-A 4-fluorosalicyclic acid derivative and process for production thereof IHARA CHEMICAL INDUSTRY CO., LTD. (JP) 2000-12-26 US disclosed
EP-0757028-B1 Process for the preparation of aromatic carbonic acid esters CLARIANT GMBH (DE) 1999-12-29 EP disclosed
US-5874608-A Process for the preparation of esters of aromatic carboxylic acid HOECHST AKTIENGESELLSCHAFT (DE) 1999-02-23 US disclosed
EP-0894784-A1 4-FLUOROSALICYLIC ACID DERIVATIVES AND PROCESS FOR PRODUCING THE SAME IHARA CHEMICAL INDUSTRY Co., Ltd. (JP) 1999-02-03 EP disclosed
US-5777181-A 2, 4, 5-trihalogeno- and 2, 3, 4, 5-tetrahalogenobenzene derivatives BAYER AKTIENGESELLSCHAFT (DE) 1998-07-07 US disclosed
EP-0811601-A1 Process for the preparation of aromatic carbonic acid esters Clariant GmbH (DE) 1997-12-10 EP disclosed
EP-0757028-A1 Process for the preparation of aromatic carbonic acid esters HOECHST AKTIENGESELLSCHAFT (DE) 1997-02-05 EP disclosed
US-5565614-A FLUORINATION BAYER AKTIENGESELLSCHAFT (DE) 1996-10-15 US disclosed
US-5530158-A CHEMICAL INTERMEDIATE FOR ANTIBACTERIALS BAYER AKTIENGESELLSCHAFT (DE) 1996-06-25 US disclosed
US-5362909-A Two stage fluorination BAYER AKTIENGESELLSCHAFT (DE) 1994-11-08 US disclosed
EP-0296479-B1 Fluorobenzoates and process for their production IHARA CHEMICAL IND CO (JP) 1994-03-30 EP disclosed
US-5200548-A Intermediates for bactericides BAYER AKTIENGESELLSCHAFT (DE) 1993-04-06 US disclosed
US-5072038-A Chemical intermediates for bactericides BAYER AKTIENGESELLSCHAFT (DE) 1991-12-10 US disclosed
US-4916253-A Fluorobenzoates and process for their production IHARA CHEMICAL INDUSTRY COMPANY, LTD. (JP) 1990-04-10 US disclosed
EP-0296479-A2 Fluorobenzoates and process for their production IHARA CHEMICAL INDUSTRY Co., Ltd. (JP) 1988-12-28 EP disclosed
EP-0164619-B1 2,4,5-TRIHALO OR 2,3,4,5-TETRAHALO BENZENE DERIVATIVES AND PROCESS FOR PRODUCING THEM BAYER AG (DE) 1988-10-12 EP disclosed